Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 68 hits in this display
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
Ki: 5.30nMAssay Description:Displacement of [3H]reserpine from human VMAT2 expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
Ki: 630nMAssay Description:Displacement of [3H]DHTB from human VMAT2 expressed in HEK293 cell membranes incubated for 90 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
IC50: 2nMpH: 8.5Assay Description:The uptake assay was performed in reaction buffer containing 140 mM K2-tartrate, 10 mM Tricine, 10 mM Tris, and 5 mM MgCl2, pH 8.5. Liposomes (1 _...More data for this Ligand-Target Pair
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
IC50: 2.5nMpH: 8.5Assay Description:The uptake assay was performed in reaction buffer containing 140 mM K2-tartrate, 10 mM Tricine, 10 mM Tris, and 5 mM MgCl2, pH 8.5. Liposomes (1 _...More data for this Ligand-Target Pair
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
IC50: 3.70nMpH: 8.5Assay Description:The uptake assay was performed in reaction buffer containing 140 mM K2-tartrate, 10 mM Tricine, 10 mM Tris, and 5 mM MgCl2, pH 8.5. Liposomes (1 _...More data for this Ligand-Target Pair
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
IC50: 3.80nMpH: 8.5Assay Description:The uptake assay was performed in reaction buffer containing 140 mM K2-tartrate, 10 mM Tricine, 10 mM Tris, and 5 mM MgCl2, pH 8.5. Liposomes (1 _...More data for this Ligand-Target Pair
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
IC50: 4.30nMpH: 8.5Assay Description:The uptake assay was performed in reaction buffer containing 140 mM K2-tartrate, 10 mM Tricine, 10 mM Tris, and 5 mM MgCl2, pH 8.5. Liposomes (1 _...More data for this Ligand-Target Pair
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
IC50: 4.5nMpH: 8.5Assay Description:The uptake assay was performed in reaction buffer containing 140 mM K2-tartrate, 10 mM Tricine, 10 mM Tris, and 5 mM MgCl2, pH 8.5. Liposomes (1 _...More data for this Ligand-Target Pair
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
IC50: 4.90nMpH: 8.5Assay Description:The uptake assay was performed in reaction buffer containing 140 mM K2-tartrate, 10 mM Tricine, 10 mM Tris, and 5 mM MgCl2, pH 8.5. Liposomes (1 _...More data for this Ligand-Target Pair
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
IC50: >50nMpH: 8.5Assay Description:The uptake assay was performed in reaction buffer containing 140 mM K2-tartrate, 10 mM Tricine, 10 mM Tris, and 5 mM MgCl2, pH 8.5. Liposomes (1 _...More data for this Ligand-Target Pair
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
IC50: >100nMpH: 8.5Assay Description:The uptake assay was performed in reaction buffer containing 140 mM K2-tartrate, 10 mM Tricine, 10 mM Tris, and 5 mM MgCl2, pH 8.5. Liposomes (1 _...More data for this Ligand-Target Pair
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
IC50: 7.00E+3nMAssay Description:Inhibition of NorA in Staphylococcus aureus 1199B assessed as inhibition of ethidium bromide efflux dose response curve based fluorometric assayMore data for this Ligand-Target Pair
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
IC50: 8.20E+3nMAssay Description:Inhibition of norA-mediated ethidium bromide efflux in methicillin-resistant Staphylococcus aureus SA-1199B by spectrofluorometric analysisMore data for this Ligand-Target Pair
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
IC50: 9.00E+3nMAssay Description:Inhibition of Staphylococcus aureus 1199B NorA assessed as reduction in ethidium bromide efflux by fluorescence assayMore data for this Ligand-Target Pair
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
IC50: 9.20E+3nMAssay Description:Inhibition of Staphylococcus aureus SA-1199B NorA assessed as reduction in EtBr efflux measured over 5 mins by fluorescence assayMore data for this Ligand-Target Pair
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
IC50: 1.02E+4nMAssay Description:TP_TRANSPORTER: increase in dihydrofluorescein intracellular accumulation (dihydrofluorescein: 1 uM) in SK-E2 cells (expressing BSEP)More data for this Ligand-Target Pair
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
BDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
Kd: 8nMAssay Description:Binding affinity to human VMAT2 expressed in HEK293 cell membranes by scintillation counting method based saturation binding assayMore data for this Ligand-Target Pair
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