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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
9
hits in this display
Target
Solute carrier family 15 member 2
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM50350470
(CEFEPIME | Maxipime)
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Affinity Data
Ki: 1.10E+7nM
Assay Description:
Binding affinity to human PepT2 in SKTP cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
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Target
Solute carrier family 15 member 2
(Rattus norvegicus)
Biozentrum Of The Martin-Luther-University Halle-Wittenberg
Curated by
ChEMBL
Ligand
BDBM50350470
(CEFEPIME | Maxipime)
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Affinity Data
Ki: 1.14E+7nM
Assay Description:
TP_TRANSPORTER: inhibition of Gly-Sar uptake (pH6.0) in SKPT cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
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ChEBI
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MCE
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PubMed
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Target
Solute carrier family 15 member 1
(Homo sapiens (Human))
Martin-Luther-University Halle-Wittenberg
Curated by
ChEMBL
Ligand
BDBM50350470
(CEFEPIME | Maxipime)
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Affinity Data
Ki: >3.00E+7nM
Assay Description:
Binding affinity against membrane transport protein PEPT1 in human Caco-2 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
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ChEBI
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MCE
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Article
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Target
Solute carrier family 15 member 1
(Homo sapiens (Human))
Martin-Luther-University Halle-Wittenberg
Curated by
ChEMBL
Ligand
BDBM50350470
(CEFEPIME | Maxipime)
Copy SMILES
Copy InChI
Affinity Data
Ki: >3.00E+7nM
Assay Description:
TP_TRANSPORTER: inhibition of Gly-Sar uptake (pH6.0) in Caco-2 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
ChEBI
DrugBank
MCE
KEGG
PC cid
PC sid
Patents
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In Depth
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Article
PubMed
DrugBank
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Target
Peptidoglycan D,D-transpeptidase FtsI
(Pseudomonas aeruginosa)
Johnson & Johnson Pharmaceutical Research And Development
Curated by
ChEMBL
Ligand
BDBM50350470
(CEFEPIME | Maxipime)
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Affinity Data
IC50: 208nM
Assay Description:
Inhibition of bocillin FL binding to Pseudomonas aeruginosa PAO1 penicillin-binding protein 3
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/TrEMBL
GoogleScholar
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Target
Peptidoglycan D,D-transpeptidase MrdA
(Escherichia coli)
Johnson & Johnson Pharmaceutical Research And Development
Curated by
ChEMBL
Ligand
BDBM50350470
(CEFEPIME | Maxipime)
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Affinity Data
IC50: 1.24E+3nM
Assay Description:
Inhibition of bocillin FL binding to Escherichia coli MC4100 penicillin-binding protein 2
More data for this Ligand-Target Pair
Target Info
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Target
Penicillin-binding protein 1B
(Pseudomonas aeruginosa)
Johnson & Johnson Pharmaceutical Research And Development
Curated by
ChEMBL
Ligand
BDBM50350470
(CEFEPIME | Maxipime)
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Affinity Data
IC50: 4.16E+3nM
Assay Description:
Inhibition of bocillin FL binding to Pseudomonas aeruginosa PAO1 penicillin-binding protein 1b
More data for this Ligand-Target Pair
Target Info
UniProtKB/TrEMBL
GoogleScholar
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Target
Peptidoglycan D,D-transpeptidase MrdA
(Pseudomonas aeruginosa)
Johnson & Johnson Pharmaceutical Research And Development
Curated by
ChEMBL
Ligand
BDBM50350470
(CEFEPIME | Maxipime)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.66E+4nM
Assay Description:
Inhibition of bocillin FL binding to Pseudomonas aeruginosa PAO1 penicillin-binding protein 2
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/TrEMBL
GoogleScholar
Ligand Info
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ChEBI
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MCE
KEGG
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In Depth
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Article
PubMed
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Target
Solute carrier family 22 member 5
(Homo sapiens)
Medical College Of Georgia
Curated by
ChEMBL
Ligand
BDBM50350470
(CEFEPIME | Maxipime)
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Affinity Data
IC50: 1.70E+6nM
Assay Description:
TP_TRANSPORTER: inhibition of Carnitine uptake (Carnitine: 0.02 uM) in OCTN2-expressing HeLa cells
More data for this Ligand-Target Pair
Target Info
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
Purchase
ChEBI
DrugBank
MCE
KEGG
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI