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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
7
hits in this display
Target
Dual specificity protein kinase TTK
(Homo sapiens (Human))
Guangzhou Institutes Of Biomedicine And Health
Curated by
ChEMBL
Ligand
BDBM50569979
(CHEMBL4875028)
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Affinity Data
IC50: 23nM
Assay Description:
Inhibition of recombinant full-length human TTK using MBP as substrate incubated for 40 mins in presence of [gamma33P]ATP by scintillation counting b...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
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Target
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
(Homo sapiens (Human))
Guangzhou Institutes Of Biomedicine And Health
Curated by
ChEMBL
Ligand
BDBM50569979
(CHEMBL4875028)
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Affinity Data
Kd: >1.00E+3nM
Assay Description:
Binding affinity to wild-type human partial length PIK3CD (R108 to Q1044 residues) expressed in HEK293 cells by active site-directed competition bind...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Interleukin-1 receptor-associated kinase 1
(Homo sapiens (Human))
Guangzhou Institutes Of Biomedicine And Health
Curated by
ChEMBL
Ligand
BDBM50569979
(CHEMBL4875028)
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Affinity Data
Kd: >1.00E+3nM
Assay Description:
Binding affinity to wild-type human partial length IRAK1 (R194 to S712 residues) expressed in mammalian expression system by active site-directed com...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
MAP/microtubule affinity-regulating kinase 3
(Homo sapiens (Human))
Guangzhou Institutes Of Biomedicine And Health
Curated by
ChEMBL
Ligand
BDBM50569979
(CHEMBL4875028)
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Affinity Data
Kd: 11nM
Assay Description:
Binding affinity to wild-type human full length MARK3 (M1 to L729 residues) expressed in bacterial expression system by measuring active site-directe...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Phosphatidylinositol 3-kinase C2 domain-containing subunit gamma
(Homo sapiens (Human))
Guangzhou Institutes Of Biomedicine And Health
Curated by
ChEMBL
Ligand
BDBM50569979
(CHEMBL4875028)
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Copy InChI
Affinity Data
Kd: >1.00E+3nM
Assay Description:
Binding affinity to human partial length PIK3C2G (M1 to I1446 residues) expressed in mammalian expression system by active site-directed competition ...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Dual specificity protein kinase TTK
(Homo sapiens (Human))
Guangzhou Institutes Of Biomedicine And Health
Curated by
ChEMBL
Ligand
BDBM50569979
(CHEMBL4875028)
Copy SMILES
Copy InChI
Affinity Data
Kd: 0.150nM
Assay Description:
Binding affinity to wild-type human partial length TTK (N505 to V798 residues) expressed in bacterial expression system by active site-directed compe...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Death-associated protein kinase 3
(Homo sapiens (Human))
Guangzhou Institutes Of Biomedicine And Health
Curated by
ChEMBL
Ligand
BDBM50569979
(CHEMBL4875028)
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Affinity Data
Kd: 13nM
Assay Description:
Binding affinity to wild-type human partial length DAPK3 (M1 to A277 residues) expressed in bacterial expression system by measuring active site-dire...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI