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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 22 hits in this display   

TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of recombinant AXL (unknown origin) using poly (Glu,Tyr) 4:1 as substrate incubated for 60 mins in presence of ATP by ELISAMore data for this Ligand-Target Pair
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TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataIC50:  27nMAssay Description:Inhibition of CSF1R (unknown origin)More data for this Ligand-Target Pair
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TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataIC50:  151nMAssay Description:Inhibition of KIT (unknown origin)More data for this Ligand-Target Pair
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TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataIC50:  156nMAssay Description:Inhibition of FLT3 (unknown origin)More data for this Ligand-Target Pair
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TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PDGFRB (unknown origin)More data for this Ligand-Target Pair
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TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataKd:  19nMAssay Description:Binding affinity to FLT4 (unknown origin) assessed as dissociation constant by competition binding assayMore data for this Ligand-Target Pair
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TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataKd:  2.60nMAssay Description:Binding affinity to KIT (unknown origin) assessed as dissociation constant by competition binding assayMore data for this Ligand-Target Pair
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TargetSerine/threonine-protein kinase 10(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataKd:  880nMAssay Description:Binding affinity to LOK (unknown origin) assessed as dissociation constant by competition binding assayMore data for this Ligand-Target Pair
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TargetMitogen-activated protein kinase kinase kinase kinase 5(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to MAP4K5 (unknown origin) assessed as dissociation constant by competition binding assayMore data for this Ligand-Target Pair
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TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataKd:  560nMAssay Description:Binding affinity to MERTK (unknown origin) assessed as dissociation constant by competition binding assayMore data for this Ligand-Target Pair
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TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to MET (unknown origin) assessed as dissociation constant by competition binding assayMore data for this Ligand-Target Pair
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TargetMacrophage-stimulating protein receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to MSTIR (unknown origin) assessed as dissociation constant by competition binding assayMore data for this Ligand-Target Pair
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TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataKd:  2.30nMAssay Description:Binding affinity to PDGFRB (unknown origin) assessed as dissociation constant by competition binding assayMore data for this Ligand-Target Pair
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TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataKd:  600nMAssay Description:Binding affinity to RET (unknown origin) assessed as dissociation constant by competition binding assayMore data for this Ligand-Target Pair
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TargetTyrosine-protein kinase receptor Tie-1(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataKd:  0.740nMAssay Description:Binding affinity to TIE1 (unknown origin) assessed as dissociation constant by competition binding assayMore data for this Ligand-Target Pair
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TargetAngiopoietin-1 receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataKd:  950nMAssay Description:Binding affinity to TIE2 (unknown origin) assessed as dissociation constant by competition binding assayMore data for this Ligand-Target Pair
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TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataKd:  2.5nMAssay Description:Binding affinity to FLT3 (unknown origin) assessed as dissociation constant by competition binding assayMore data for this Ligand-Target Pair
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TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataKd:  14nMAssay Description:Binding affinity to FLT1 (unknown origin) assessed as dissociation constant by competition binding assayMore data for this Ligand-Target Pair
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TargetEphrin type-B receptor 6(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to EPHB6 (unknown origin) assessed as dissociation constant by competition binding assayMore data for this Ligand-Target Pair
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TargetEpithelial discoidin domain-containing receptor 1(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to DDR1 (unknown origin) assessed as dissociation constant by competition binding assayMore data for this Ligand-Target Pair
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TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataKd:  29nMAssay Description:Binding affinity to CSF1R (unknown origin) assessed as dissociation constant by competition binding assayMore data for this Ligand-Target Pair
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TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50588796(CHEMBL5197792)
Affinity DataKd:  0.260nMAssay Description:Binding affinity to AXL (unknown origin) assessed as dissociation constant by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails PubMed