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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
11
hits in this display
Target
G-protein coupled receptor 35
(Homo sapiens (Human))
University Of Bonn
Curated by
ChEMBL
Ligand
BDBM50436001
(CHEMBL2392174 | CHEMBL2425818)
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Affinity Data
Ki: 5.20nM
Assay Description:
Displacement of [3H]PSB-13253 from human recombinant GPR35 exprssed in CHO cells by liquid scintillation counting analysis
Checked by Author
More data for this Ligand-Target Pair
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Target
G-protein coupled receptor 55
(Homo sapiens (Human))
University Of Bonn
Curated by
ChEMBL
Ligand
BDBM50436001
(CHEMBL2392174 | CHEMBL2425818)
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Affinity Data
IC50: 2.17E+4nM
Assay Description:
Antagonist activity at human GPR55 expressed in CHO cells assessed as inhibition of lysophosphotidylinositol-induced beta-arrestin recruitment preinc...
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Target
G-protein coupled receptor 35
(Homo sapiens (Human))
University Of Bonn
Curated by
ChEMBL
Ligand
BDBM50436001
(CHEMBL2392174 | CHEMBL2425818)
Copy SMILES
Copy InChI
Affinity Data
Kd: 115nM
Assay Description:
Binding affinity to human recombinant GPR35 expressed in CHO cells by scintillation counting analysis in absence of MgCl2, NaCl, CaCl2
Checked by Author
More data for this Ligand-Target Pair
Target Info
PDB
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KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
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CHEMBL
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In Depth
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Article
PubMed
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Target
G-protein coupled receptor 35
(Homo sapiens (Human))
University Of Bonn
Curated by
ChEMBL
Ligand
BDBM50436001
(CHEMBL2392174 | CHEMBL2425818)
Copy SMILES
Copy InChI
Affinity Data
Kd: 5.30nM
Assay Description:
Binding affinity to human recombinant GPR35 expressed in CHO cells after 150 mins by liquid scintillation counting analysis
Checked by Author
More data for this Ligand-Target Pair
Target Info
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KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
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CHEMBL
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In Depth
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Article
PubMed
Copy BDB DOI
Target
G-protein coupled receptor 35
(Homo sapiens (Human))
University Of Bonn
Curated by
ChEMBL
Ligand
BDBM50436001
(CHEMBL2392174 | CHEMBL2425818)
Copy SMILES
Copy InChI
Affinity Data
Kd: 5.90nM
Assay Description:
Competitive binding affinity to human recombinant GPR35 expressed in CHO cells by scintillation counting analysis in presence of CaCl2
Checked by Author
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
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CHEMBL
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PC sid
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In Depth
Details
Article
PubMed
Copy BDB DOI
Target
G-protein coupled receptor 35
(Homo sapiens (Human))
University Of Bonn
Curated by
ChEMBL
Ligand
BDBM50436001
(CHEMBL2392174 | CHEMBL2425818)
Copy SMILES
Copy InChI
Affinity Data
EC50: 12nM
Assay Description:
Agonist activity at human GPR35 expressed in CHO-K1 cells after 90 mins by beta-arrestin 2 recruitment assay
More data for this Ligand-Target Pair
Target Info
PDB
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KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
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CHEMBL
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PC sid
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In Depth
Details
Article
PubMed
Copy BDB DOI
Target
G-protein coupled receptor 35
(Homo sapiens (Human))
University Of Bonn
Curated by
ChEMBL
Ligand
BDBM50436001
(CHEMBL2392174 | CHEMBL2425818)
Copy SMILES
Copy InChI
Affinity Data
Kd: 5.70nM
Assay Description:
Competitive binding affinity to human recombinant GPR35 expressed in CHO cells by scintillation counting analysis in presence of MgCl2
Checked by Author
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
G-protein coupled receptor 35
(Homo sapiens (Human))
University Of Bonn
Curated by
ChEMBL
Ligand
BDBM50436001
(CHEMBL2392174 | CHEMBL2425818)
Copy SMILES
Copy InChI
Affinity Data
EC50: 22nM
Assay Description:
Agonist activity at human GPR35b expressed in CHO cells assessed as induction of beta-arrestin recruitment after 90 mins by beta-galactosidase report...
More data for this Ligand-Target Pair
Target Info
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GoogleScholar
Ligand Info
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CHEMBL
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In Depth
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Article
PubMed
Copy BDB DOI
Target
G protein-coupled receptor GPR35
(Rattus norvegicus)
University Of Bonn
Curated by
ChEMBL
Ligand
BDBM50436001
(CHEMBL2392174 | CHEMBL2425818)
Copy SMILES
Copy InChI
Affinity Data
EC50: 1.40E+3nM
Assay Description:
Agonist activity at rat GPR35 expressed in CHO cells assessed as induction of beta-arrestin recruitment after 90 mins by beta-galactosidase reporter ...
More data for this Ligand-Target Pair
Target Info
KEGG
UniProtKB/TrEMBL
GoogleScholar
Ligand Info
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CHEMBL
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PC sid
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In Depth
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Article
PubMed
Copy BDB DOI
Target
G-protein coupled receptor 35
(Homo sapiens (Human))
University Of Bonn
Curated by
ChEMBL
Ligand
BDBM50436001
(CHEMBL2392174 | CHEMBL2425818)
Copy SMILES
Copy InChI
Affinity Data
EC50: 12nM
Assay Description:
Agonist activity at human GPR35 expressed in CHO cells assessed as induction of beta-arrestin recruitment after 90 mins by beta-galactosidase reporte...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
G-protein coupled receptor 35
(Homo sapiens (Human))
University Of Bonn
Curated by
ChEMBL
Ligand
BDBM50436001
(CHEMBL2392174 | CHEMBL2425818)
Copy SMILES
Copy InChI
Affinity Data
EC50: 12nM
Assay Description:
Agonist activity at human GPR35 expressed in CHO cells assessed as induction of beta-arrestin recruitment after 90 mins by beta-galactosidase reporte...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI