Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 26 hits in this display
ADAMTS5(Rattus norvegicus (Rat))Galapagos
US Patent
BDBM379557(US9926281, Compound 36)
BDBM379557(US9926281, Compound 36)
IC50: 34nMAssay Description:Inhibition of human recombinant ADAMTS-5 assessed as cleavage of fluorescent substrate using FAM-TBIS-1 by biochemical assayMore data for this Ligand-Target Pair
BDBM379557(US9926281, Compound 36)
BDBM379557(US9926281, Compound 36)
BDBM379557(US9926281, Compound 36)
BDBM379557(US9926281, Compound 36)
BDBM379557(US9926281, Compound 36)
BDBM379557(US9926281, Compound 36)
BDBM379557(US9926281, Compound 36)
BDBM379557(US9926281, Compound 36)
BDBM379557(US9926281, Compound 36)
BDBM379557(US9926281, Compound 36)
BDBM379557(US9926281, Compound 36)
BDBM379557(US9926281, Compound 36)
BDBM379557(US9926281, Compound 36)
BDBM379557(US9926281, Compound 36)
BDBM379557(US9926281, Compound 36)
BDBM379557(US9926281, Compound 36)
BDBM379557(US9926281, Compound 36)
BDBM379557(US9926281, Compound 36)
BDBM379557(US9926281, Compound 36)
BDBM379557(US9926281, Compound 36)
BDBM379557(US9926281, Compound 36)
BDBM379557(US9926281, Compound 36)
BDBM379557(US9926281, Compound 36)
BDBM379557(US9926281, Compound 36)