TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: >1.00E+3nM ΔG°: >-34.2kJ/molepH: 7.0 T: 2°CAssay Description:PTP activity was assayed using p-nitrophenyl phosphate (pNPP) as a substrate in DMG buffer (50 mM DMG, pH 7.0, 1 mM EDTA, 150 mM NaCl, 2 mM DTT, 0.1 ...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: 1.30E+3nMAssay Description:Inhibition of LAR (unknown origin)More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: 1.60E+3nMAssay Description:Inhibition of LAR (unknown origin) using pNPP as substrate preincubated for 5 mins followed by substrate addition measured for 20 mins by spectrophot...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: >3.00E+3nMAssay Description:Inhibitory activity against SH-domain containing phosphotyrosine phosphatase-2 (Tyrosine phosphatase SHP2) was determinedMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: 2.14E+4nM ΔG°: -26.4kJ/molepH: 7.4 T: 2°CAssay Description:The reaction was started by addition of pNPP substrate, and reaction progress was monitored at 405 nm. The initial rate data collected was used for d...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: >3.00E+4nMAssay Description:Inhibitory potency of the compound against LARMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: >3.00E+4nMAssay Description:Inhibitory potency of the compound against LARMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: >3.00E+4nMAssay Description:Inhibitory potency of the compound against LARMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: 5.00E+4nMpH: 5.5Assay Description:Inhibitory effect against protein-tyrosine phosphatase Lar, using p-nitrophenyl phosphate as substrate at pH 5.5.More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: 5.00E+4nMpH: 5.5Assay Description:Inhibitory effect against protein-tyrosine phosphatase Lar, using p-nitrophenyl phosphate as substrate at pH 5.5.More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: 6.80E+4nMAssay Description:Inhibition of PTPRFMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: 9.00E+4nMpH: 5.5Assay Description:Inhibitory effect against protein-tyrosine phosphatase Lar, using p-nitrophenyl phosphate as substrate at pH 5.5.More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: 9.00E+4nMpH: 5.5Assay Description:Inhibitory effect against protein-tyrosine phosphatase Lar, using p-nitrophenyl phosphate as substrate at pH 5.5.More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: 9.60E+4nMAssay Description:Inhibitory activity against SH-domain containing phosphotyrosine phosphatase-2 (Tyrosine phosphatase SHP2) was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+5nMAssay Description:Inhibition of rat recombinant LAR expressed in Escherichia coli assessed as inhibition constant using pNPP as substrate incubated for 5 mins by liqui...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human LARMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: 1.10E+5nMpH: 5.5Assay Description:Inhibitory effect against protein-tyrosine phosphatase Lar, using p-nitrophenyl phosphate as substrate at pH 5.5.More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: 1.13E+5nMpH: 5.5Assay Description:Inhibitory effect against protein-tyrosine phosphatase Lar, using p-nitrophenyl phosphate as substrate at pH 5.5.More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: 1.30E+5nMAssay Description:Non-covalent inhibition of LAR (unknown origin) using DiFMUP as substrate incubated for 15 to 120 mins followed by substrate addition at pH 6.5 by st...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: 1.30E+5nMAssay Description:Non-covalent inhibition of LAR (unknown origin) using DiFMUP as substrate incubated for 15 to 120 mins followed by substrate addition at pH 6.5 by st...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: 1.60E+5nMpH: 5.5Assay Description:Inhibitory effect against protein-tyrosine phosphatase Lar, using p-nitrophenyl phosphate as substrate at pH 5.5.More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: 1.65E+5nMpH: 5.5Assay Description:Inhibitory effect against protein-tyrosine phosphatase Lar, using p-nitrophenyl phosphate as substrate at pH 5.5.More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: 1.76E+5nMAssay Description:Inhibition of PTPRFMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: 3.20E+5nMAssay Description:Inhibition of PTPRFMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: 3.60E+5nMAssay Description:Inhibition of human LAR using pNPP as substrate after 5 mins by spectrophotometric plate reader analysisMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: 3.60E+5nMpH: 5.5Assay Description:Inhibitory effect against protein-tyrosine phosphatase Lar, using p-nitrophenyl phosphate as substrate at pH 5.5.More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: 3.60E+5nMAssay Description:Inhibition of PTPRFMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: 3.90E+5nMAssay Description:Inhibition of human LAR using pNPP as substrate after 5 mins by spectrophotometric plate reader analysisMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: 4.00E+5nMpH: 5.5Assay Description:Inhibitory effect against protein-tyrosine phosphatase Lar, using p-nitrophenyl phosphate as substrate at pH 5.5.More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: 4.10E+5nMAssay Description:Inhibition of PTPRFMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: 4.10E+5nMpH: 5.5Assay Description:Inhibitory effect against protein-tyrosine phosphatase Lar, using p-nitrophenyl phosphate as substrate at pH 5.5.More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: 4.20E+5nMpH: 5.5Assay Description:Inhibitory effect against protein-tyrosine phosphatase Lar, using p-nitrophenyl phosphate as substrate at pH 5.5.More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: 4.20E+5nMAssay Description:Inhibition of PTPRFMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: 4.50E+5nMpH: 5.5Assay Description:Inhibitory effect against protein-tyrosine phosphatase Lar, using p-nitrophenyl phosphate as substrate at pH 5.5.More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: 4.50E+5nMAssay Description:Inhibition of PTPRFMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: 4.50E+5nMAssay Description:Inhibition of LAR (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: >5.00E+5nMAssay Description:Inhibition of PTPRFMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: >5.00E+5nMAssay Description:Inhibition of human recombinant LARMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: >5.00E+5nMAssay Description:Inhibition of human recombinant LARMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: 5.50E+5nMpH: 5.5Assay Description:Inhibitory effect against protein-tyrosine phosphatase Lar, using p-nitrophenyl phosphate as substrate at pH 5.5.More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: 5.50E+5nMAssay Description:Inhibition of PTPRFMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: 7.00E+5nMpH: 5.5Assay Description:Inhibitory effect against protein-tyrosine phosphatase Lar, using p-nitrophenyl phosphate as substrate at pH 5.5.More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: 9.00E+5nMpH: 5.5Assay Description:Inhibitory effect against protein-tyrosine phosphatase Lar, using p-nitrophenyl phosphate as substrate at pH 5.5.More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: >9.00E+5nMAssay Description:Inhibition of human LAR using pNPP as substrate after 5 mins by spectrophotometric plate reader analysisMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of human recombinant LARMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of PTPRFMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of PTPRFMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of PTPRFMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: 1.10E+6nMAssay Description:Inhibition of PTPRFMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: 2.00E+6nMpH: 5.5Assay Description:Inhibitory effect against protein-tyrosine phosphatase Lar, using p-nitrophenyl phosphate as substrate at pH 5.5.More data for this Ligand-Target Pair