Report error Found 2850 Enz. Inhib. hit(s) with Target = 'Cathepsin B'
Affinity DataKi: 0.0110nM ΔG°: -65.1kJ/molepH: 6.0 T: 37°CAssay Description:Enzyme was equilibrated in 0.1 M phosphate buffer, pH 6.0 at 37 °C. All compounds were prepared in DMSO. Various concentrations of compounds we...More data for this Ligand-Target Pair
Affinity DataKi: 0.0200nMAssay Description:Competitive inhibition of goat brain cathepsin BMore data for this Ligand-Target Pair
Affinity DataKi: 0.0770nMAssay Description:Inhibition constant against human cathepsin B in fluorescence assay using Cbz-Phe-Arg-AMCMore data for this Ligand-Target Pair
Affinity DataKi: 0.0870nMAssay Description:Kinetic parameter (Ki 1/min) was evaluated for the inactivation of cathepsin BMore data for this Ligand-Target Pair
Affinity DataKi: 0.0940nMAssay Description:Inhibition of bovine cathepsin BMore data for this Ligand-Target Pair
Affinity DataKi: 0.113nM ΔG°: -59.1kJ/molepH: 6.0 T: 37°CAssay Description:Enzyme was equilibrated in 0.1 M phosphate buffer, pH 6.0 at 37 °C. All compounds were prepared in DMSO. Various concentrations of compounds we...More data for this Ligand-Target Pair
Affinity DataKi: 0.140nMAssay Description:Inhibition of bovine cathepsin BMore data for this Ligand-Target Pair
Affinity DataKi: 0.141nM ΔG°: -58.5kJ/molepH: 6.0 T: 37°CAssay Description:Enzyme was equilibrated in 0.1 M phosphate buffer, pH 6.0 at 37 °C. All compounds were prepared in DMSO. Various concentrations of compounds we...More data for this Ligand-Target Pair
Affinity DataKi: 0.146nM ΔG°: -58.4kJ/molepH: 6.0 T: 37°CAssay Description:Enzyme was equilibrated in 0.1 M phosphate buffer, pH 6.0 at 37 °C. All compounds were prepared in DMSO. Various concentrations of compounds we...More data for this Ligand-Target Pair
Affinity DataKi: 0.180nM ΔG°: -57.9kJ/molepH: 6.0 T: 37°CAssay Description:Enzyme was equilibrated in 0.1 M phosphate buffer, pH 6.0 at 37 °C. All compounds were prepared in DMSO. Various concentrations of compounds we...More data for this Ligand-Target Pair
Affinity DataKi: 0.211nM ΔG°: -57.4kJ/molepH: 6.0 T: 37°CAssay Description:Enzyme was equilibrated in 0.1 M phosphate buffer, pH 6.0 at 37 °C. All compounds were prepared in DMSO. Various concentrations of compounds we...More data for this Ligand-Target Pair
Affinity DataKi: 0.227nM ΔG°: -57.3kJ/molepH: 6.0 T: 37°CAssay Description:Enzyme was equilibrated in 0.1 M phosphate buffer, pH 6.0 at 37 °C. All compounds were prepared in DMSO. Various concentrations of compounds we...More data for this Ligand-Target Pair
Affinity DataKi: 0.25nMAssay Description:Inhibition constant against human cathepsin B in fluorescence assay using Cbz-Phe-Arg-AMCMore data for this Ligand-Target Pair
Affinity DataKi: 0.360nMAssay Description:Inhibition of human recombinant cathepsin B after 30 mins by spectrophotometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.380nMAssay Description:Inhibition of human recombinant cathepsin B after 30 mins by spectrophotometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.406nMAssay Description:Inhibition of human cathepsin B using Z-Arg-Arg-pNA chromogenic substrate fluorogenic substrate incubated for 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 0.430nMAssay Description:Inhibition of human recombinant cathepsin B after 30 mins by spectrophotometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.448nM ΔG°: -55.5kJ/molepH: 6.0 T: 37°CAssay Description:Enzyme was equilibrated in 0.1 M phosphate buffer, pH 6.0 at 37 °C. All compounds were prepared in DMSO. Various concentrations of compounds we...More data for this Ligand-Target Pair
Affinity DataKi: 0.455nM ΔG°: -55.5kJ/molepH: 6.0 T: 37°CAssay Description:Enzyme was equilibrated in 0.1 M phosphate buffer, pH 6.0 at 37 °C. All compounds were prepared in DMSO. Various concentrations of compounds we...More data for this Ligand-Target Pair
Affinity DataKi: 0.459nMAssay Description:Inhibition of human cathepsin B using Z-Arg-Arg-pNA chromogenic substrate fluorogenic substrate incubated for 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 0.480nMAssay Description:Inhibition of human recombinant cathepsin B after 30 mins by spectrophotometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.650nMAssay Description:Inhibition of human recombinant cathepsin B after 30 mins by spectrophotometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.668nM ΔG°: -54.5kJ/molepH: 6.0 T: 37°CAssay Description:Enzyme was equilibrated in 0.1 M phosphate buffer, pH 6.0 at 37 °C. All compounds were prepared in DMSO. Various concentrations of compounds we...More data for this Ligand-Target Pair
Affinity DataKi: 0.680nMAssay Description:Inhibition of human recombinant cathepsin B after 30 mins by spectrophotometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.690nMAssay Description:Inhibition of human liver cathepsin B using Z-Phe-Arg-AMC as substrate incubated for 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.880nMAssay Description:Inhibition of human recombinant cathepsin B after 30 mins by spectrophotometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Equilibrium dissociation constant of the compound for the inhibition of human cathepsin B was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Inhibition constant against human cathepsin B in fluorescence assay using Cbz-Phe-Arg-AMCMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Inhibition of human recombinant cathepsin B after 30 mins by spectrophotometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Inhibition of human recombinant cathepsin B after 30 mins by spectrophotometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Inhibitory activity of the compound against cathepsin BMore data for this Ligand-Target Pair
Affinity DataKi: 1.95nM ΔG°: -51.7kJ/molepH: 6.0 T: 37°CAssay Description:Enzyme was equilibrated in 0.1 M phosphate buffer, pH 6.0 at 37 °C. All compounds were prepared in DMSO. Various concentrations of compounds we...More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:In vitro inhibitory activity against beta-1 adrenergic receptor determined as pA2 in guinea pig atriaMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of human liver cathepsin B using Z-Phe-Arg-AMC as substrate incubated for 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of human cathepsin BMore data for this Ligand-Target Pair
Affinity DataKi: 2nMpH: 5.5Assay Description:A fluorometric high-throughput assay for activity against cathepsin B was performed in 96-well microtiter plates. The assay were performed in Dynate...More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of human liver cathepsin BMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Inhibition of human recombinant cathepsin B after 30 mins by spectrophotometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Inhibition of human recombinant cathepsin B after 30 mins by spectrophotometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Inhibition of human recombinant cathepsin B after 30 mins by spectrophotometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.87nM ΔG°: -50.7kJ/molepH: 6.0 T: 37°CAssay Description:Enzyme was equilibrated in 0.1 M phosphate buffer, pH 6.0 at 37 °C. All compounds were prepared in DMSO. Various concentrations of compounds we...More data for this Ligand-Target Pair
Affinity DataKi: 3.36nMAssay Description:Inhibition of cathepsin BMore data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Inhibition of human cathepsin B using Z-Arg-Arg-pNA chromogenic substrate fluorogenic substrate incubated for 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Inhibitory activity of the compound against cathepsin BMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Inhibitory activity against cathepsin B receptor in human liverMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Inhibitory activity of the compound against cathepsin BMore data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:Inhibition of human recombinant cathepsin B after 30 mins by spectrophotometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:Inhibition of human cathepsin BMore data for this Ligand-Target Pair
Affinity DataKi: 4.70nMpH: 5.5Assay Description:A fluorometric high-throughput assay for activity against cathepsin B was performed in 96-well microtiter plates. The assay were performed in Dynate...More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibitory activity of the compound against cathepsin BMore data for this Ligand-Target Pair
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