TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataKi: >4.00E+5nMAssay Description:Displacement of FAM- labeled YAP1 peptide from TEAD2 (217 to 447 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as inhi...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4/Isoform 5 of Transcriptional coactivator [50-100](Homo sapiens)
Genentech
US Patent
Genentech
US Patent
Affinity DataIC50: 10nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4/Isoform 5 of Transcriptional coactivator [50-100](Homo sapiens)
Genentech
US Patent
Genentech
US Patent
Affinity DataIC50: 10nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4/Isoform 5 of Transcriptional coactivator [50-100](Homo sapiens)
Genentech
US Patent
Genentech
US Patent
Affinity DataIC50: 10nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4/Isoform 5 of Transcriptional coactivator [50-100](Homo sapiens)
Genentech
US Patent
Genentech
US Patent
Affinity DataIC50: 10nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4/Isoform 5 of Transcriptional coactivator [50-100](Homo sapiens)
Genentech
US Patent
Genentech
US Patent
Affinity DataIC50: 10nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4/Isoform 5 of Transcriptional coactivator [50-100](Homo sapiens)
Genentech
US Patent
Genentech
US Patent
Affinity DataIC50: 10nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4/Isoform 5 of Transcriptional coactivator [50-100](Homo sapiens)
Genentech
US Patent
Genentech
US Patent
Affinity DataIC50: 20nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4/Isoform 5 of Transcriptional coactivator [50-100](Homo sapiens)
Genentech
US Patent
Genentech
US Patent
Affinity DataIC50: 30nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4/Isoform 5 of Transcriptional coactivator [50-100](Homo sapiens)
Genentech
US Patent
Genentech
US Patent
Affinity DataIC50: 50nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4/Isoform 5 of Transcriptional coactivator [50-100](Homo sapiens)
Genentech
US Patent
Genentech
US Patent
Affinity DataIC50: 50nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4/Isoform 5 of Transcriptional coactivator [50-100](Homo sapiens)
Genentech
US Patent
Genentech
US Patent
Affinity DataIC50: 60nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4/Isoform 5 of Transcriptional coactivator [50-100](Homo sapiens)
Genentech
US Patent
Genentech
US Patent
Affinity DataIC50: 70nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4/Isoform 5 of Transcriptional coactivator [50-100](Homo sapiens)
Genentech
US Patent
Genentech
US Patent
Affinity DataIC50: 80nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4/Isoform 5 of Transcriptional coactivator [50-100](Homo sapiens)
Genentech
US Patent
Genentech
US Patent
Affinity DataIC50: 130nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-4(Homo sapiens)
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataIC50: 240nMAssay Description:Table 2-3: His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid p...More data for this Ligand-Target Pair