Compile Data Set for Download or QSAR
maximum 50k data
Found 7 of ki for monomerid = 50387827
TargetNischarin(RAT)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50387827(CHEMBL2058635)
Affinity DataKi:  0.178nMAssay Description:Displacement of [125I]PIC from Imidazoline-1 receptor in rat PC12 cell membrane incubated for 30 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50387827(CHEMBL2058635)
Affinity DataKi:  0.200nMAssay Description:Displacement of [125I] PIC from I1 imidazoline receptor in rat PC12 cells after 45 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50387827(CHEMBL2058635)
Affinity DataKi:  0.219nMAssay Description:Displacement of [3H]paraiodoclonidine from imidazoline I1 receptor in rat PC12 cells after 30 mins by gamma counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50387827(CHEMBL2058635)
Affinity DataKi: >2.50E+3nMAssay Description:Displacement of [3H]RX821002 from human alpha2 adrenoceptor expressed in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50387827(CHEMBL2058635)
Affinity DataKi:  2.57E+3nMAssay Description:Displacement of [3H]RX821001 from human alpha2A adrenoceptor expressed in CHO cells after 60 mins by gamma counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50387827(CHEMBL2058635)
Affinity DataKi:  4.17E+3nMAssay Description:Displacement of [3H]RX821001 from human alpha2B adrenoceptor expressed in CHO cells after 60 mins by gamma counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50387827(CHEMBL2058635)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]RX821001 from human alpha2C adrenoceptor expressed in CHO cells after 60 mins by gamma counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed