Compile Data Set for Download or QSAR
maximum 50k data
Found 8 of ki for monomerid = 50600748
TargetAdenosine receptor A2a(Homo sapiens (Human))
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50600748(CHEMBL5176737)
Affinity DataKi:  0.0810nMAssay Description:Displacement of [3H]ZM241385 from human A2AAR expressed in HEK293 cells membrane assessed as inhibition constant preincubated for 5 mins followed by ...More data for this Ligand-Target Pair
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TargetAdenosine receptor A2a(Homo sapiens (Human))
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50600748(CHEMBL5176737)
Affinity DataKi:  0.302nMAssay Description:Displacement of [3H]ZM241385 from human A2AAR expressed in HEK293 cells membrane assessed as inhibition constant preincubated for 5 mins followed by ...More data for this Ligand-Target Pair
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TargetAdenosine receptor A1(Homo sapiens (Human))
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50600748(CHEMBL5176737)
Affinity DataKi:  7.40nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in HEK293 cells membrane assessed as inhibition constant preincubated for 5 mins followed by [3H]...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A1(Homo sapiens (Human))
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50600748(CHEMBL5176737)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in HEK293 cells membrane assessed as inhibition constant preincubated for 5 mins followed by [3H]...More data for this Ligand-Target Pair
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TargetAdenosine receptor A2b(Homo sapiens (Human))
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50600748(CHEMBL5176737)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]DPCPX from human A2BAR expressed in HEK293 cells membrane assessed as inhibition constant preincubated for 5 mins followed by [3H...More data for this Ligand-Target Pair
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TargetAdenosine receptor A2b(Homo sapiens (Human))
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50600748(CHEMBL5176737)
Affinity DataKi:  97nMAssay Description:Displacement of [3H]DPCPX from human A2BAR expressed in HEK293 cells membrane assessed as inhibition constant preincubated for 5 mins followed by [3H...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A3(Homo sapiens (Human))
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50600748(CHEMBL5176737)
Affinity DataKi:  1.26E+3nMAssay Description:Displacement of [3H]HEMADO from human A3AR expressed in CHO-K1 cells membrane assessed as inhibition constant preincubated for 5 mins followed by [3H...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50600748(CHEMBL5176737)
Affinity DataKi:  3.05E+3nMAssay Description:Displacement of [3H]HEMADO from human A3AR expressed in CHO-K1 cells membrane assessed as inhibition constant preincubated for 5 mins followed by [3H...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed