TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataKi: 501nMAssay Description:Binding affinity to CK1a1 (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataKi: 650nMAssay Description:Binding affinity to CK1a1 (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition of CK1 (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition of CK1 (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition of CK1 (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataKi: >6.92E+3nMAssay Description:Inhibition of CK1alpha1More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataKi: 3.83E+4nMAssay Description:Inhibition of casein kinase 1Checked by AuthorMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataKi: 3.83E+4nM ΔG°: -6.12kcal/moleT: 2°CAssay Description:Protein kinase C, cAMP dependent protein kinase, cGMP dependent protein kinase and myosin light chain kinase activity were measure under conditions d...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataKi: 6.07E+4nM ΔG°: -5.85kcal/moleT: 2°CAssay Description:Protein kinase C, cAMP dependent protein kinase, cGMP dependent protein kinase and myosin light chain kinase activity were measure under conditions d...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataKi: 8.00E+4nMAssay Description:Inhibition of casein kinase 1Checked by AuthorMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of human CK1-alpha1More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of Ck1alpha1More data for this Ligand-Target Pair