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Found 4 Enz. Inhib. hit(s) with all data for entry = 50010890
TargetHTH-type quorum-sensing regulator RhlR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Korea University

Curated by ChEMBL
LigandPNGBDBM50543115(CHEMBL4642992)
Affinity DataIC50:  2.60E+4nMAssay Description:Antagonist activity at Pseudomonas aeruginosa RhlR expressed in Escherichia coli DH5alpha incubated for 1.5 hrs by luminescence reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type quorum-sensing regulator RhlR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Korea University

Curated by ChEMBL
LigandPNGBDBM50543114(CHEMBL4632586)
Affinity DataIC50:  8.60E+4nMAssay Description:Antagonist activity at Pseudomonas aeruginosa RhlR expressed in Escherichia coli DH5alpha incubated for 1.5 hrs by luminescence reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type quorum-sensing regulator RhlR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Korea University

Curated by ChEMBL
LigandPNGBDBM50210051(CHEMBL3883439)
Affinity DataIC50:  2.18E+5nMAssay Description:Antagonist activity at Pseudomonas aeruginosa RhlR expressed in Escherichia coli DH5alpha incubated for 1.5 hrs by luminescence reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type quorum-sensing regulator RhlR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Korea University

Curated by ChEMBL
LigandPNGBDBM50275147(6-Gingerol | BDBM50317427 | CHEMBL446043 | Gingero...)
Affinity DataIC50:  9.45E+5nMAssay Description:Antagonist activity at Pseudomonas aeruginosa RhlR expressed in Escherichia coli DH5alpha incubated for 1.5 hrs by luminescence reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed