Compile Data Set for Download or QSAR
maximum 50k data
Found 41 Enz. Inhib. hit(s) with all data for entry = 50010930
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50543539(CHEMBL4638480)
Affinity DataIC50:  0.760nMAssay Description:Inhibition of DPP4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50543537(CHEMBL4649180)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of DPP4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50543538(CHEMBL4632896)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of DPP4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50543532(CHEMBL4641140)
Affinity DataIC50:  2.80nMAssay Description:Inhibition of recombinant human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition by florescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50543534(CHEMBL4647761)
Affinity DataIC50:  5.80nMAssay Description:Inhibition of DPP4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50543536(CHEMBL4642801)
Affinity DataIC50:  6nMAssay Description:Inhibition of DPP4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50543541(CHEMBL4638352)
Affinity DataIC50:  12nMAssay Description:Inhibition of DPP4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50338518(1-((3S,4S)-4-amino-1-(4-(3,3-difluoropyrrolidin-1-...)
Affinity DataIC50:  23nMAssay Description:Inhibition of DPP4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50543533(CHEMBL4636081)
Affinity DataIC50:  29nMAssay Description:Inhibition of recombinant human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50543509(CHEMBL4636119)
Affinity DataIC50:  70nMAssay Description:Inhibition of PTP1B (unknown origin) using p-NPP as substrate after 0.5 hrsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50543540(CHEMBL4647956)
Affinity DataIC50:  247nMAssay Description:Inhibition of DPP4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50543511(CHEMBL4641922)
Affinity DataIC50:  880nMAssay Description:Inhibition of PTP1B (unknown origin) by fluorometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50543514(CHEMBL4642505)
Affinity DataIC50:  1.88E+3nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50543515(CHEMBL4636382)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50543510(CHEMBL4637354)
Affinity DataIC50:  3.33E+3nMAssay Description:Inhibition of PTP1B (unknown origin) by fluorometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mizoram University

Curated by ChEMBL
LigandPNGBDBM11695((2S)-1-{2-[(3-hydroxyadamantan-1-yl)amino]acetyl}p...)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of DPP4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50543517(CHEMBL4635202)
Affinity DataIC50:  7.31E+3nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50543516(CHEMBL4639896)
Affinity DataIC50:  8.73E+3nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50462424(CHEMBL4246951)
Affinity DataIC50:  2.81E+4nMAssay Description:Inhibition of recombinant human DPP4 using Gly-Pro-AMC as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50543513(CHEMBL4634743)
Affinity DataIC50:  4.36E+4nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50543512(CHEMBL4648808)
Affinity DataIC50:  4.40E+4nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens)
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50543527(CHEMBL4647832)
Affinity DataEC50:  179nMAssay Description:Agonist activity at GPR120 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens)
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50543528(CHEMBL4638249)
Affinity DataEC50:  110nMAssay Description:Agonist activity at GPR120 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens)
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50543529(CHEMBL4641735)
Affinity DataEC50:  270nMAssay Description:Agonist activity at GPR120 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens)
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50543530(CHEMBL4646784)
Affinity DataEC50:  6nMAssay Description:Agonist activity at GPR120 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens)
Mizoram University

Curated by ChEMBL
LigandPNGBDBM382129(4-(4-((4'-cyclopropyl-3,4,5,6-tetrahydro-[1,1'-bip...)
Affinity DataEC50:  50nMAssay Description:Agonist activity at GPR120 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50543520(CHEMBL4642473)
Affinity DataEC50:  33nMAssay Description:Inhibition of human SGLT2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50543531(CHEMBL4635583)
Affinity DataEC50:  270nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50543521(CHEMBL4633698)
Affinity DataEC50:  797nMAssay Description:Agonist activity at GPR40 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50543520(CHEMBL4642473)
Affinity DataEC50:  37nMAssay Description:Inhibition of human SGLT1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50543519(CHEMBL4642324)
Affinity DataEC50:  71nMAssay Description:Modulation of GPR40 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50543535(CHEMBL4632639)
Affinity DataEC50:  1.20nMAssay Description:Inhibition of DPP4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50085584(5-(4-{2-[1-(6-Phenyl-pyridin-3-yl)-eth-(E)-ylidene...)
Affinity DataEC50:  190nMAssay Description:Agonist activity at PPARgamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50543518(CHEMBL4639604)
Affinity DataEC50:  8.90nMAssay Description:Agonist activity at PPARgamma (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens)
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50543526(CHEMBL4646553)
Affinity DataEC50:  61nMAssay Description:Agonist activity at GPR120 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens)
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50543525(CHEMBL4639009)
Affinity DataEC50:  45nMAssay Description:Agonist activity at GPR120 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens)
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50543524(CHEMBL4637969)
Affinity DataEC50:  6nMAssay Description:Agonist activity at GPR120 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens)
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50543519(CHEMBL4642324)
Affinity DataEC50:  71nMAssay Description:Modulation of GPR120 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50543522(CHEMBL4638816)
Affinity DataEC50:  648nMAssay Description:Agonist activity at GPR40 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50339460(3-[4-(Biphenyl-3-ylmethoxy)phenyl]propanoic Acid |...)
Affinity DataEC50:  75nMAssay Description:Agonist activity at GPR40 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens)
Mizoram University

Curated by ChEMBL
LigandPNGBDBM50543523(CHEMBL4642294)
Affinity DataEC50:  220nMAssay Description:Modulation of GPR120 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed