Affinity DataIC50: 0.760nMAssay Description:Inhibition of DPP4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Inhibition of DPP4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Inhibition of DPP4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.80nMAssay Description:Inhibition of recombinant human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition by florescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.80nMAssay Description:Inhibition of DPP4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of DPP4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of DPP4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of DPP4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Inhibition of recombinant human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate additionMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Mizoram University
Curated by ChEMBL
Mizoram University
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibition of PTP1B (unknown origin) using p-NPP as substrate after 0.5 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 247nMAssay Description:Inhibition of DPP4 (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Mizoram University
Curated by ChEMBL
Mizoram University
Curated by ChEMBL
Affinity DataIC50: 880nMAssay Description:Inhibition of PTP1B (unknown origin) by fluorometric assayMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Mizoram University
Curated by ChEMBL
Mizoram University
Curated by ChEMBL
Affinity DataIC50: 1.88E+3nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Mizoram University
Curated by ChEMBL
Mizoram University
Curated by ChEMBL
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Mizoram University
Curated by ChEMBL
Mizoram University
Curated by ChEMBL
Affinity DataIC50: 3.33E+3nMAssay Description:Inhibition of PTP1B (unknown origin) by fluorometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of DPP4 (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Mizoram University
Curated by ChEMBL
Mizoram University
Curated by ChEMBL
Affinity DataIC50: 7.31E+3nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Mizoram University
Curated by ChEMBL
Mizoram University
Curated by ChEMBL
Affinity DataIC50: 8.73E+3nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.81E+4nMAssay Description:Inhibition of recombinant human DPP4 using Gly-Pro-AMC as substrate after 30 minsMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Mizoram University
Curated by ChEMBL
Mizoram University
Curated by ChEMBL
Affinity DataIC50: 4.36E+4nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Mizoram University
Curated by ChEMBL
Mizoram University
Curated by ChEMBL
Affinity DataIC50: 4.40E+4nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 179nMAssay Description:Agonist activity at GPR120 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 110nMAssay Description:Agonist activity at GPR120 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 270nMAssay Description:Agonist activity at GPR120 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 6nMAssay Description:Agonist activity at GPR120 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Agonist activity at GPR120 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 33nMAssay Description:Inhibition of human SGLT2More data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Mizoram University
Curated by ChEMBL
Mizoram University
Curated by ChEMBL
Affinity DataEC50: 270nMAssay Description:Agonist activity at human GPR119More data for this Ligand-Target Pair
Affinity DataEC50: 797nMAssay Description:Agonist activity at GPR40 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 37nMAssay Description:Inhibition of human SGLT1More data for this Ligand-Target Pair
Affinity DataEC50: 71nMAssay Description:Modulation of GPR40 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 1.20nMAssay Description:Inhibition of DPP4 (unknown origin)More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Mizoram University
Curated by ChEMBL
Mizoram University
Curated by ChEMBL
Affinity DataEC50: 190nMAssay Description:Agonist activity at PPARgamma (unknown origin)More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Mizoram University
Curated by ChEMBL
Mizoram University
Curated by ChEMBL
Affinity DataEC50: 8.90nMAssay Description:Agonist activity at PPARgamma (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 61nMAssay Description:Agonist activity at GPR120 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 45nMAssay Description:Agonist activity at GPR120 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 6nMAssay Description:Agonist activity at GPR120 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 71nMAssay Description:Modulation of GPR120 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 648nMAssay Description:Agonist activity at GPR40 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 75nMAssay Description:Agonist activity at GPR40 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 220nMAssay Description:Modulation of GPR120 (unknown origin)More data for this Ligand-Target Pair