BindingDB PrimarySearch_ki

Found 38 Enz. Inhib. hit(s) with all data for entry = 50012261

Serine/threonine-protein kinase PAK 1(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50148931(CHEMBL3770186)

Ki: 0.0230nMAssay Description:Inhibition of full length recombinant human N-terminal GST/His6-tagged PAK1 expressed in sf9 insect cells using tetra LRRWSLG as substrate preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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3D Structure (crystal)

Serine/threonine-protein kinase PAK 1(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50555982(CHEMBL4758500)

IC50: 9.80nMAssay Description:Inhibition of full length recombinant human N-terminal GST/His6-tagged PAK1 expressed in sf9 insect cells using tetra LRRWSLG as substrate preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Serine/threonine-protein kinase PAK 4(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM101536(CHEMBL3128043 | US8530494, 203 | US8530652, 114 | ...)

IC50: 15nMAssay Description:Inhibition of PAK4 (unknown origin)More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Serine/threonine-protein kinase PAK 1(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50555981(CHEMBL4794004)

IC50: 16nMAssay Description:Inhibition of full length recombinant human N-terminal GST/His6-tagged PAK1 expressed in sf9 insect cells using tetra LRRWSLG as substrate preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Details Article PubMed

Serine/threonine-protein kinase PAK 1(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50555968(CHEMBL4742230)

IC50: 16nMAssay Description:Inhibition of full length recombinant human N-terminal GST/His6-tagged PAK1 expressed in sf9 insect cells using tetra LRRWSLG as substrate preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Details Article PubMed

Serine/threonine-protein kinase PAK 1(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50555983(CHEMBL4787358)

IC50: 21nMAssay Description:Inhibition of full length recombinant human N-terminal GST/His6-tagged PAK1 expressed in sf9 insect cells using tetra LRRWSLG as substrate preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Details Article PubMed

Serine/threonine-protein kinase PAK 1(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50555980(CHEMBL4784979)

IC50: 22nMAssay Description:Inhibition of full length recombinant human N-terminal GST/His6-tagged PAK1 expressed in sf9 insect cells using tetra LRRWSLG as substrate preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Details Article PubMed

Serine/threonine-protein kinase PAK 1(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50555970(CHEMBL4781551)

IC50: 34nMAssay Description:Inhibition of full length recombinant human N-terminal GST/His6-tagged PAK1 expressed in sf9 insect cells using tetra LRRWSLG as substrate preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Details Article PubMed

Serine/threonine-protein kinase PAK 4(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM101536(CHEMBL3128043 | US8530494, 203 | US8530652, 114 | ...)

IC50: 38nMAssay Description:Inhibition of full length recombinant human N-terminal GST/His6-tagged PAK4 expressed in baculovirus infected sf9 insect cells using tetra LRRWSLG as...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Serine/threonine-protein kinase PAK 1(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM101536(CHEMBL3128043 | US8530494, 203 | US8530652, 114 | ...)

IC50: 39nMAssay Description:Inhibition of PAK1 (unknown origin)More data for this Ligand-Target Pair

PDB Reactome pathway
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Serine/threonine-protein kinase PAK 1(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50555979(CHEMBL4784560)

IC50: 42nMAssay Description:Inhibition of full length recombinant human N-terminal GST/His6-tagged PAK1 expressed in sf9 insect cells using tetra LRRWSLG as substrate preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Details Article PubMed

Serine/threonine-protein kinase PAK 1(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50555972(CHEMBL4748552)

IC50: 45nMAssay Description:Inhibition of full length recombinant human N-terminal GST/His6-tagged PAK1 expressed in sf9 insect cells using tetra LRRWSLG as substrate preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Details Article PubMed

Serine/threonine-protein kinase PAK 1(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM101536(CHEMBL3128043 | US8530494, 203 | US8530652, 114 | ...)

IC50: 52nMAssay Description:Inhibition of full length recombinant human N-terminal GST/His6-tagged PAK1 expressed in sf9 insect cells using tetra LRRWSLG as substrate preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

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Serine/threonine-protein kinase PAK 1(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50555965(CHEMBL4799349)

IC50: 52nMAssay Description:Inhibition of full length recombinant human N-terminal GST/His6-tagged PAK1 expressed in sf9 insect cells using tetra LRRWSLG as substrate preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Details Article PubMed

Serine/threonine-protein kinase PAK 1(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50555973(CHEMBL4750093)

IC50: 66nMAssay Description:Inhibition of full length recombinant human N-terminal GST/His6-tagged PAK1 expressed in sf9 insect cells using tetra LRRWSLG as substrate preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

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Serine/threonine-protein kinase PAK 1(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50555974(CHEMBL4764182)

IC50: 71nMAssay Description:Inhibition of full length recombinant human N-terminal GST/His6-tagged PAK1 expressed in sf9 insect cells using tetra LRRWSLG as substrate preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Details Article PubMed

Serine/threonine-protein kinase PAK 1(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50555984(CHEMBL4764341)

IC50: 92nMAssay Description:Inhibition of full length recombinant human N-terminal GST/His6-tagged PAK1 expressed in sf9 insect cells using tetra LRRWSLG as substrate preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Details Article PubMed

Serine/threonine-protein kinase PAK 1(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50555978(CHEMBL4755754)

IC50: 143nMAssay Description:Inhibition of full length recombinant human N-terminal GST/His6-tagged PAK1 expressed in sf9 insect cells using tetra LRRWSLG as substrate preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Details Article PubMed

Serine/threonine-protein kinase PAK 1(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50555964(CHEMBL4790872)

IC50: 159nMAssay Description:Inhibition of full length recombinant human N-terminal GST/His6-tagged PAK1 expressed in sf9 insect cells using tetra LRRWSLG as substrate preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Details Article PubMed

Serine/threonine-protein kinase PAK 1(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50555967(CHEMBL4789576)

IC50: 229nMAssay Description:Inhibition of full length recombinant human N-terminal GST/His6-tagged PAK1 expressed in sf9 insect cells using tetra LRRWSLG as substrate preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Details Article PubMed

Serine/threonine-protein kinase PAK 1(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50555969(CHEMBL4763427)

IC50: 330nMAssay Description:Inhibition of full length recombinant human N-terminal GST/His6-tagged PAK1 expressed in sf9 insect cells using tetra LRRWSLG as substrate preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Details Article PubMed

Serine/threonine-protein kinase PAK 1(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50555971(CHEMBL4782048)

IC50: 590nMAssay Description:Inhibition of full length recombinant human N-terminal GST/His6-tagged PAK1 expressed in sf9 insect cells using tetra LRRWSLG as substrate preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Details Article PubMed

Serine/threonine-protein kinase PAK 1(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50555977(CHEMBL4794451)

IC50: 744nMAssay Description:Inhibition of full length recombinant human N-terminal GST/His6-tagged PAK1 expressed in sf9 insect cells using tetra LRRWSLG as substrate preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Details Article PubMed

Serine/threonine-protein kinase PAK 1(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50555966(CHEMBL4783727)

IC50: 777nMAssay Description:Inhibition of full length recombinant human N-terminal GST/His6-tagged PAK1 expressed in sf9 insect cells using tetra LRRWSLG as substrate preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Details Article PubMed

Serine/threonine-protein kinase PAK 1(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50555963(CHEMBL4748736)

IC50: 5.00E+3nMAssay Description:Inhibition of full length recombinant human N-terminal GST/His6-tagged PAK1 expressed in sf9 insect cells using tetra LRRWSLG as substrate preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Details Article PubMed

Serine/threonine-protein kinase PAK 1(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50555963(CHEMBL4748736)

IC50: 5.00E+3nMAssay Description:Inhibition of PAK1 (unknown origin)More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Details Article PubMed

Serine/threonine-protein kinase PAK 1(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50555976(CHEMBL4752794)

IC50: >1.00E+4nMAssay Description:Inhibition of full length recombinant human N-terminal GST/His6-tagged PAK1 expressed in sf9 insect cells using tetra LRRWSLG as substrate preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Details Article PubMed

Serine/threonine-protein kinase PAK 4(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50555972(CHEMBL4748552)

IC50: >1.00E+4nMAssay Description:Inhibition of full length recombinant human N-terminal GST/His6-tagged PAK4 expressed in baculovirus infected sf9 insect cells using tetra LRRWSLG as...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Details Article PubMed

Serine/threonine-protein kinase PAK 4(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50555982(CHEMBL4758500)

IC50: >1.00E+4nMAssay Description:Inhibition of full length recombinant human N-terminal GST/His6-tagged PAK4 expressed in baculovirus infected sf9 insect cells using tetra LRRWSLG as...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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Serine/threonine-protein kinase PAK 4(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50555968(CHEMBL4742230)

IC50: >1.00E+4nMAssay Description:Inhibition of full length recombinant human N-terminal GST/His6-tagged PAK4 expressed in baculovirus infected sf9 insect cells using tetra LRRWSLG as...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Details Article PubMed

Serine/threonine-protein kinase PAK 1(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50555975(CHEMBL4753834)

IC50: >1.00E+4nMAssay Description:Inhibition of full length recombinant human N-terminal GST/His6-tagged PAK1 expressed in sf9 insect cells using tetra LRRWSLG as substrate preincubat...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Details Article PubMed

Serine/threonine-protein kinase PAK 4(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50555970(CHEMBL4781551)

IC50: >1.00E+4nMAssay Description:Inhibition of full length recombinant human N-terminal GST/His6-tagged PAK4 expressed in baculovirus infected sf9 insect cells using tetra LRRWSLG as...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Details Article PubMed

Potassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50555972(CHEMBL4748552)

IC50: 1.60E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Potassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50555968(CHEMBL4742230)

IC50: 2.10E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Potassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50555982(CHEMBL4758500)

IC50: 4.11E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Potassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM101536(CHEMBL3128043 | US8530494, 203 | US8530652, 114 | ...)

IC50: 4.21E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Potassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50555970(CHEMBL4781551)

IC50: 8.23E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Potassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

PNG

BDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)

IC50: 9.04E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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