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Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50015754
TargetTranscription factor 4(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50589362(CHEMBL5181203)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of His-tagged beta-catenin (134 to 668 residues)/CM-5 sensor chip immobilized N-terminal GST-tagged TCF4 interaction (unknown origin) prei...More data for this Ligand-Target Pair
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TargetCatenin beta-1(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50589357(CHEMBL5178667)
Affinity DataKd:  53nMAssay Description:Binding affinity to human beta-catenin (134 to 665 residues) expressed in Escherichia coli BL21 assessed as dissociation constant incubated for 45 mi...More data for this Ligand-Target Pair
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TargetCatenin beta-1(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50589358(CHEMBL5178520)
Affinity DataKd:  123nMAssay Description:Binding affinity to full-length recombinant beta-catenin (unknown origin) assessed as dissociation constant by fluorescence polarisation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetCatenin beta-1(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50589359(CHEMBL5205469)
Affinity DataKd:  5nMAssay Description:Binding affinity to human beta-catenin (129 to 780 residues) expressed in Escherichia coli Rosetta blue assessed as dissociation constant using fluor...More data for this Ligand-Target Pair
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TargetCatenin beta-1(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50589360(CHEMBL5180356)
Affinity DataKd:  5nMAssay Description:Binding affinity to human beta-catenin (129 to 780 residues) expressed in Escherichia coli Rosetta blue assessed as dissociation constant using fluor...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetCatenin beta-1(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50589364(CHEMBL5186135)
Affinity DataKd:  91nMAssay Description:Binding affinity to full-length beta-catenin (1 to 781 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as dissociation c...More data for this Ligand-Target Pair
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TargetCatenin beta-1(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50014132(CHEMBL2323032)
Affinity DataKd:  530nMAssay Description:Binding affinity to human beta-catenin (138 to 686 residues) assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCatenin beta-1(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50589361(CHEMBL5181546)
Affinity DataKd:  420nMAssay Description:Binding affinity to beta-catenin (unknown origin) assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCatenin beta-1(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50589362(CHEMBL5181203)
Affinity DataKd:  5.80E+5nMAssay Description:Binding affinity to CM-5 sensor chip immobilized His-tagged beta-catenin (134 to 668 residues) (unknown origin) expressed in Escherichia coli BL21 as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCatenin beta-1(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50589363(CHEMBL5191201)
Affinity DataKd:  156nMAssay Description:Binding affinity to full-length beta-catenin (1 to 781 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as dissociation c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetCatenin beta-1(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50589356(CHEMBL5194459)
Affinity DataKd:  13nMAssay Description:Binding affinity to human beta-catenin (134 to 665 residues) expressed in Escherichia coli BL21 assessed as dissociation constant incubated for 45 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetCatenin beta-1(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50436058(CHEMBL254381 | PNU-74654 | US9738628, Compound PNU...)
Affinity DataKd:  450nMAssay Description:Binding affinity to beta-catenin (134 to 671 residues) (unknown origin) expressed in Escherichia coli BL21 assessed as dissociation constant by isoth...More data for this Ligand-Target Pair
In DepthDetails PubMed