Report error Found 80 Enz. Inhib. hit(s) with all data for entry = 50016875
TargetHistone-arginine methyltransferase CARM1(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 3.20nMAssay Description:Inhibition of human full length recombinant GST-tagged PRMT4 (2 to 608 residues) using histone H3 as substrate incubated for 20 mins in presence of [...More data for this Ligand-Target Pair
TargetHistone-arginine methyltransferase CARM1(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 8.40nMAssay Description:Inhibition of human full length recombinant GST-tagged PRMT4 (2 to 608 residues) using histone H3 as substrate incubated for 20 mins in presence of [...More data for this Ligand-Target Pair
TargetHistone-arginine methyltransferase CARM1(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 9.70nMAssay Description:Inhibition of human full length recombinant GST-tagged PRMT4 (2 to 608 residues) using histone H3 as substrate incubated for 20 mins in presence of [...More data for this Ligand-Target Pair
TargetHistone-arginine methyltransferase CARM1(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 43nMAssay Description:Inhibition of PRMT4 (unknown origin)More data for this Ligand-Target Pair
TargetHistone-arginine methyltransferase CARM1(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 68nMAssay Description:Inhibition of human full length recombinant GST-tagged PRMT4 (2 to 608 residues) using histone H3 as substrate incubated for 20 mins in presence of [...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 5(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 113nMAssay Description:Inhibition of human full length recombinant FLAG-tagged PRMT5 (2 to 637 residues) using histone H2A as substrate incubated for 20 mins in presence of...More data for this Ligand-Target Pair
TargetHistone-arginine methyltransferase CARM1(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 176nMAssay Description:Inhibition of human full length recombinant GST-tagged PRMT4 (2 to 608 residues) using histone H3 as substrate incubated for 20 mins in presence of [...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 7(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of human full length recombinant his-tagged PRMT7 (2 to 692 residues) using GST-GAR as substrate incubated for 20 mins in presence of [3H]...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 7(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 226nMAssay Description:Inhibition of human full length recombinant his-tagged PRMT7 (2 to 692 residues) using GST-GAR as substrate incubated for 20 mins in presence of [3H]...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 7(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 320nMAssay Description:Inhibition of human full length recombinant his-tagged PRMT7 (2 to 692 residues) using GST-GAR as substrate incubated for 20 mins in presence of [3H]...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Inhibition of recombinant human PRMT1 assessed as residual activity using biotinylated histone H4 (1 to 21) as substrate incubated for 60 mins in pre...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 7(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 410nMAssay Description:Inhibition of human full length recombinant his-tagged PRMT7 (2 to 692 residues) using GST-GAR as substrate incubated for 20 mins in presence of [3H]...More data for this Ligand-Target Pair
TargetHistone-arginine methyltransferase CARM1(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 420nMAssay Description:Inhibition of human full length recombinant GST-tagged PRMT4 (2 to 608 residues) using histone H3 as substrate incubated for 20 mins in presence of [...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 7(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 550nMAssay Description:Inhibition of human full length recombinant his-tagged PRMT7 (2 to 692 residues) using GST-GAR as substrate incubated for 20 mins in presence of [3H]...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 7(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 631nMAssay Description:Inhibition of human full length recombinant his-tagged PRMT7 (2 to 692 residues) using GST-GAR as substrate incubated for 20 mins in presence of [3H]...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 5(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 778nMAssay Description:Inhibition of human full length recombinant FLAG-tagged PRMT5 (2 to 637 residues) using histone H2A as substrate incubated for 20 mins in presence of...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 835nMAssay Description:Inhibition of human full length recombinant GST-tagged PRMT1 (2 to 371 residues) using histone H4 as substrate incubated for 20 mins in presence of [...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 860nMAssay Description:Inhibition of human full length recombinant GST-tagged PRMT1 (2 to 371 residues) using histone H4 as substrate incubated for 20 mins in presence of [...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of recombinant human PRMT1 assessed as residual activity using biotinylated histone H4 (1 to 21) as substrate incubated for 60 mins in pre...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 8(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 1.41E+3nMAssay Description:Inhibition of human full length recombinant his-tagged PRMT8 (61 to 394 residues) using histone H4 as substrate incubated for 20 mins in presence of ...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 5(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 1.46E+3nMAssay Description:Inhibition of human full length recombinant FLAG-tagged PRMT5 (2 to 637 residues) using histone H2A as substrate incubated for 20 mins in presence of...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of recombinant human PRMT1 assessed as residual activity using biotinylated histone H4 (1 to 21) as substrate incubated for 60 mins in pre...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 7(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 1.68E+3nMAssay Description:Inhibition of human full length recombinant his-tagged PRMT7 (2 to 692 residues) using GST-GAR as substrate incubated for 20 mins in presence of [3H]...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 6(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 1.75E+3nMAssay Description:Inhibition of human full length recombinant GST-tagged PRMT6 (2 to 375 residues) using GST-GAR as substrate incubated for 20 mins in presence of [3H]...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of human full length recombinant GST-tagged PRMT1 (2 to 371 residues) using histone H4 as substrate incubated for 20 mins in presence of [...More data for this Ligand-Target Pair
TargetHistone-arginine methyltransferase CARM1(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of PRMT4 (unknown origin)More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 8(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 1.95E+3nMAssay Description:Inhibition of human full length recombinant his-tagged PRMT8 (61 to 394 residues) using histone H4 as substrate incubated for 20 mins in presence of ...More data for this Ligand-Target Pair
TargetHistone-arginine methyltransferase CARM1(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 2.14E+3nMAssay Description:Inhibition of human full length recombinant GST-tagged PRMT4 (2 to 608 residues) using histone H3 as substrate incubated for 20 mins in presence of [...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of human full length recombinant GST-tagged PRMT1 (2 to 371 residues) using histone H4 as substrate incubated for 20 mins in presence of [...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 5(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of human full length recombinant FLAG-tagged PRMT5 (2 to 637 residues) using histone H2A as substrate incubated for 20 mins in presence of...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 5(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 3.38E+3nMAssay Description:Inhibition of human full length recombinant FLAG-tagged PRMT5 (2 to 637 residues) using histone H2A as substrate incubated for 20 mins in presence of...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of recombinant human PRMT1 assessed as residual activity using biotinylated histone H4 (1 to 21) as substrate incubated for 60 mins in pre...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 8(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 3.82E+3nMAssay Description:Inhibition of human full length recombinant his-tagged PRMT8 (61 to 394 residues) using histone H4 as substrate incubated for 20 mins in presence of ...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 3(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 4.05E+3nMAssay Description:Inhibition of human full length recombinant GST his-tagged PRMT3 (2 to 531 residues) using histone H4 as substrate incubated for 20 mins in presence ...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 6(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 4.34E+3nMAssay Description:Inhibition of human full length recombinant GST-tagged PRMT6 (2 to 375 residues) using GST-GAR as substrate incubated for 20 mins in presence of [3H]...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 7(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 4.68E+3nMAssay Description:Inhibition of human full length recombinant his-tagged PRMT7 (2 to 692 residues) using GST-GAR as substrate incubated for 20 mins in presence of [3H]...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 4.86E+3nMAssay Description:Inhibition of human full length recombinant GST-tagged PRMT1 (2 to 371 residues) using histone H4 as substrate incubated for 20 mins in presence of [...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 8(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 5.84E+3nMAssay Description:Inhibition of human full length recombinant his-tagged PRMT8 (61 to 394 residues) using histone H4 as substrate incubated for 20 mins in presence of ...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 8(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 5.87E+3nMAssay Description:Inhibition of human full length recombinant his-tagged PRMT8 (61 to 394 residues) using histone H4 as substrate incubated for 20 mins in presence of ...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 8(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of human full length recombinant his-tagged PRMT8 (61 to 394 residues) using histone H4 as substrate incubated for 20 mins in presence of ...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 8(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 8.29E+3nMAssay Description:Inhibition of human full length recombinant his-tagged PRMT8 (61 to 394 residues) using histone H4 as substrate incubated for 20 mins in presence of ...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 8.46E+3nMAssay Description:Inhibition of human full length recombinant GST-tagged PRMT1 (2 to 371 residues) using histone H4 as substrate incubated for 20 mins in presence of [...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 9.30E+3nMAssay Description:Inhibition of recombinant human PRMT1 assessed as residual activity using biotinylated histone H4 (1 to 21) as substrate incubated for 60 mins in pre...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 3(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 1.05E+4nMAssay Description:Inhibition of human full length recombinant GST his-tagged PRMT3 (2 to 531 residues) using histone H4 as substrate incubated for 20 mins in presence ...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 1.17E+4nMAssay Description:Inhibition of human full length recombinant GST-tagged PRMT1 (2 to 371 residues) using histone H4 as substrate incubated for 20 mins in presence of [...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 3(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 1.22E+4nMAssay Description:Inhibition of human full length recombinant GST his-tagged PRMT3 (2 to 531 residues) using histone H4 as substrate incubated for 20 mins in presence ...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 3(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 1.24E+4nMAssay Description:Inhibition of human full length recombinant GST his-tagged PRMT3 (2 to 531 residues) using histone H4 as substrate incubated for 20 mins in presence ...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 3(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 1.33E+4nMAssay Description:Inhibition of human full length recombinant GST his-tagged PRMT3 (2 to 531 residues) using histone H4 as substrate incubated for 20 mins in presence ...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 1.37E+4nMAssay Description:Inhibition of recombinant human PRMT1 assessed as residual activity using biotinylated histone H4 (1 to 21) as substrate incubated for 60 mins in pre...More data for this Ligand-Target Pair
TargetHistone-arginine methyltransferase CARM1(Human)
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Institut De G£N£Tique Et De Biologie Mol£Culaire Et Cellulaire
Curated by ChEMBL
Affinity DataIC50: 1.38E+4nMAssay Description:Inhibition of human full length recombinant GST-tagged PRMT4 (2 to 608 residues) using histone H3 as substrate incubated for 20 mins in presence of [...More data for this Ligand-Target Pair