Affinity DataKi: 2.02E+3nMAssay Description:Antagonist activity at adrenergic Alpha-1D receptor in rat aortaMore data for this Ligand-Target Pair
Affinity DataKi: 4.62E+3nMAssay Description:Antagonist activity at adrenergic Alpha-1D receptor in rat aortaMore data for this Ligand-Target Pair
Affinity DataKi: 1.34E+4nMAssay Description:Antagonist activity at adrenergic alpha1A receptor in rat tail arteryMore data for this Ligand-Target Pair
Affinity DataIC50: 256nMAssay Description:Inhibition of human recombinant FAAHMore data for this Ligand-Target Pair
Affinity DataIC50: 282nMAssay Description:Inhibition of human recombinant FAAHMore data for this Ligand-Target Pair
Affinity DataIC50: 319nMAssay Description:Inhibition of human recombinant FAAHMore data for this Ligand-Target Pair
Affinity DataIC50: 319nMAssay Description:Inhibition of human recombinant MGLMore data for this Ligand-Target Pair
Affinity DataIC50: 319nMAssay Description:Inhibition of human recombinant FAAHMore data for this Ligand-Target Pair
Affinity DataIC50: 368nMAssay Description:Inhibition of rat brain FAAHMore data for this Ligand-Target Pair
Affinity DataIC50: 495nMAssay Description:Antagonist activity at human adenosine A1 receptor expressed in CHO FlpIn cells assessed as inhibition of of N(6)-(R-phenylisopropyl)adenosine-induce...More data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+3nMAssay Description:Antagonist activity at histamine H3 receptor in electrically-stimulated guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+3nMAssay Description:Antagonist activity at histamine H3 receptor in electrically-stimulated guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:Antagonist activity at adrenergic alpha1A receptor in rat tail arteryMore data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:Antagonist activity at adrenergic Alpha-1B receptor in guinea pig spleenMore data for this Ligand-Target Pair
Affinity DataIC50: 5.40E+3nMAssay Description:Antagonist activity at adrenergic Alpha-1B receptor in guinea pig spleenMore data for this Ligand-Target Pair
Affinity DataIC50: 6.70E+3nMAssay Description:Antagonist activity at adrenergic alpha1A receptor in rat tail arteryMore data for this Ligand-Target Pair
Affinity DataIC50: 8.10E+3nMAssay Description:Antagonist activity at histamine H3 receptor in electrically-stimulated guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+4nMAssay Description:Antagonist activity at human adenosine A1 receptor expressed in CHO FlpIn cells assessed as inhibition of of N(6)-(R-phenylisopropyl)adenosine-induce...More data for this Ligand-Target Pair
Affinity DataIC50: 3.32E+4nMAssay Description:Inhibition of human recombinant MGLMore data for this Ligand-Target Pair
Affinity DataIC50: 3.32E+4nMAssay Description:Antagonist activity at oxytocin receptor in rat uterine strips assessed as inhibition of oxytocin-induced contractionMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40E+4nMAssay Description:Antagonist activity at human adenosine A1 receptor expressed in CHO FlpIn cells assessed as inhibition of of N(6)-(R-phenylisopropyl)adenosine-induce...More data for this Ligand-Target Pair
Affinity DataIC50: 4.04E+4nMAssay Description:Inhibition of human recombinant MGLMore data for this Ligand-Target Pair
Affinity DataIC50: 4.50E+4nMAssay Description:Antagonist activity at adrenergic Alpha-1B receptor in guinea pig spleenMore data for this Ligand-Target Pair
Affinity DataIC50: 5.10E+4nMAssay Description:Antagonist activity at histamine H3 receptor in electrically-stimulated guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 7.40E+4nMAssay Description:Antagonist activity at adrenergic Alpha-1B receptor in guinea pig spleenMore data for this Ligand-Target Pair
Affinity DataIC50: 8.90E+4nMAssay Description:Antagonist activity at adrenergic Alpha-1B receptor in guinea pig spleenMore data for this Ligand-Target Pair
Affinity DataIC50: 9.50E+4nMAssay Description:Antagonist activity at adrenergic Alpha-1B receptor in guinea pig spleenMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at adrenergic alpha1A receptor in rat tail arteryMore data for this Ligand-Target Pair
Affinity DataIC50: 1.02E+5nMAssay Description:Antagonist activity at adrenergic alpha1A receptor in rat tail arteryMore data for this Ligand-Target Pair
Affinity DataIC50: 1.05E+5nMAssay Description:Antagonist activity at adrenergic alpha1A receptor in rat tail arteryMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+5nMAssay Description:Antagonist activity at adrenergic Alpha-1B receptor in guinea pig spleenMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+5nMAssay Description:Antagonist activity at adrenergic Alpha-1B receptor in guinea pig spleenMore data for this Ligand-Target Pair
Affinity DataIC50: 1.53E+5nMAssay Description:Antagonist activity at adrenergic alpha1A receptor in rat tail arteryMore data for this Ligand-Target Pair
Affinity DataIC50: 1.57E+5nMAssay Description:Antagonist activity at adrenergic Alpha-1B receptor in guinea pig spleenMore data for this Ligand-Target Pair
Affinity DataIC50: 1.77E+5nMAssay Description:Antagonist activity at adrenergic Alpha-1B receptor in guinea pig spleenMore data for this Ligand-Target Pair
Affinity DataIC50: 1.84E+5nMAssay Description:Antagonist activity at adrenergic Alpha-1B receptor in guinea pig spleenMore data for this Ligand-Target Pair
Affinity DataIC50: 1.84E+5nMAssay Description:Antagonist activity at adrenergic alpha1A receptor in rat tail arteryMore data for this Ligand-Target Pair
Affinity DataIC50: 1.87E+5nMAssay Description:Antagonist activity at adrenergic alpha1A receptor in rat tail arteryMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+5nMAssay Description:Antagonist activity at adrenergic alpha1A receptor in rat tail arteryMore data for this Ligand-Target Pair
Affinity DataEC50: 7.00E+4nMAssay Description:Antagonist activity at adrenergic Alpha-1B receptor in guinea pig spleenMore data for this Ligand-Target Pair
Affinity DataEC50: 7.10E+3nMAssay Description:Antagonist activity at adrenergic alpha1A receptor in rat tail arteryMore data for this Ligand-Target Pair
Affinity DataEC50: 7.10E+3nMAssay Description:Antagonist activity at adrenergic alpha1A receptor in rat tail arteryMore data for this Ligand-Target Pair
Affinity DataEC50: 1.03E+4nMAssay Description:Antagonist activity at oxytocin receptor in rat uterine strips assessed as inhibition of oxytocin-induced contractionMore data for this Ligand-Target Pair
Affinity DataEC50: 4.60E+5nMAssay Description:Antagonist activity at histamine H3 receptor in electrically-stimulated guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 4.04E+5nMAssay Description:Antagonist activity at histamine H3 receptor in electrically-stimulated guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 7.60E+5nMAssay Description:Antagonist activity at histamine H3 receptor in electrically-stimulated guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 3.10E+3nMAssay Description:Antagonist activity at histamine H3 receptor in electrically-stimulated guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 8.90E+4nMAssay Description:Antagonist activity at histamine H3 receptor in electrically-stimulated guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 2.30E+5nMAssay Description:Antagonist activity at histamine H3 receptor in electrically-stimulated guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 2.70E+5nMAssay Description:Antagonist activity at histamine H3 receptor in electrically-stimulated guinea pig ileumMore data for this Ligand-Target Pair