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Found 18 Enz. Inhib. hit(s) with all data for entry = 50018669
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM220664(US10633379, Compound Y | US9296741, 253)
Affinity DataKi:  1.20nMAssay Description:Binding affinity to BDR4- BD2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM220664(US10633379, Compound Y | US9296741, 253)
Affinity DataKi:  22nMAssay Description:Binding affinity to BDR4-BD1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50591847(CHEMBL5194033)
Affinity DataKi:  77nMAssay Description:Binding affinity to human BRD4 BD1 assessed as inhibition constant incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50591847(CHEMBL5194033)
Affinity DataKi:  718nMAssay Description:Binding affinity to human BRD4 BD2 assessed as inhibition constant incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50158615(Ischemin)
Affinity DataKi:  1.09E+4nMAssay Description:Inhibition of BRD4 BD1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50158615(Ischemin)
Affinity DataKi:  1.97E+4nMAssay Description:Inhibition of BRD4 BD2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50610939(CHEMBL5288200)
Affinity DataIC50:  130nMAssay Description:Inhibition of his 6 tagged BRD4 D1 (unknown origin) expressed in Escherichia coli BL21 (DE3) by fluorescence anisotropy assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))TBA
LigandPNGBDBM50103503(CHEMBL2393130 | US11117865, Compound RVX-208)
Affinity DataIC50:  510nMAssay Description:Binding affinity to BRD3 BD2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))TBA
LigandPNGBDBM50103503(CHEMBL2393130 | US11117865, Compound RVX-208)
Affinity DataIC50:  8.70E+4nMAssay Description:Binding affinity to BRD3 BD1 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))TBA
LigandPNGBDBM50610939(CHEMBL5288200)
Affinity DataKd:  1.90E+3nMAssay Description:Binding affinity to p38 alpha (unknown origin) assessed as dissociation constant by DiscoverX kinomescan methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))TBA
LigandPNGBDBM50099333(2-(3,5-Dimethyl-phenoxy)-4-[5-(4-fluoro-phenyl)-3-...)
Affinity DataKd:  0.470nMAssay Description:Binding affinity to p38 alpha (unknown origin) assessed as dissociation constant by DiscoverX kinomescan methodMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50148603(CHEMBL3770724)
Affinity DataKd:  3.40E+3nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin) assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 2(Homo sapiens (Human))TBA
LigandPNGBDBM50407714(CHEMBL5269983)
Affinity DataKd:  931nMAssay Description:Binding affinity to BDR2-BD1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50593635(CHEMBL5205867)
Affinity DataKd:  2nMAssay Description:Binding affinity to BDR4- BD2 (unknown origin) assessed as dissociation constant by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))TBA
LigandPNGBDBM50407714(CHEMBL5269983)
Affinity DataKd:  14nMAssay Description:Binding affinity to BDR2- BD2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))TBA
LigandPNGBDBM50593635(CHEMBL5205867)
Affinity DataKd:  6nMAssay Description:Binding affinity to BDR2- BD2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50593635(CHEMBL5205867)
Affinity DataKd:  301nMAssay Description:Binding affinity to BDR4-BD1 (unknown origin) assessed as dissociation constant by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))TBA
LigandPNGBDBM50593635(CHEMBL5205867)
Affinity DataKd:  490nMAssay Description:Binding affinity to BDR2-BD1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed