Affinity DataKi: 1.20nMAssay Description:Binding affinity to BDR4- BD2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Binding affinity to BDR4-BD1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 77nMAssay Description:Binding affinity to human BRD4 BD1 assessed as inhibition constant incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 718nMAssay Description:Binding affinity to human BRD4 BD2 assessed as inhibition constant incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.09E+4nMAssay Description:Inhibition of BRD4 BD1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.97E+4nMAssay Description:Inhibition of BRD4 BD2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition of his 6 tagged BRD4 D1 (unknown origin) expressed in Escherichia coli BL21 (DE3) by fluorescence anisotropy assayMore data for this Ligand-Target Pair
Affinity DataIC50: 510nMAssay Description:Binding affinity to BRD3 BD2 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.70E+4nMAssay Description:Binding affinity to BRD3 BD1 (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
Affinity DataKd: 1.90E+3nMAssay Description:Binding affinity to p38 alpha (unknown origin) assessed as dissociation constant by DiscoverX kinomescan methodMore data for this Ligand-Target Pair
Affinity DataKd: 0.470nMAssay Description:Binding affinity to p38 alpha (unknown origin) assessed as dissociation constant by DiscoverX kinomescan methodMore data for this Ligand-Target Pair
Affinity DataKd: 3.40E+3nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin) assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 931nMAssay Description:Binding affinity to BDR2-BD1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKd: 2nMAssay Description:Binding affinity to BDR4- BD2 (unknown origin) assessed as dissociation constant by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKd: 14nMAssay Description:Binding affinity to BDR2- BD2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKd: 6nMAssay Description:Binding affinity to BDR2- BD2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKd: 301nMAssay Description:Binding affinity to BDR4-BD1 (unknown origin) assessed as dissociation constant by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKd: 490nMAssay Description:Binding affinity to BDR2-BD1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair