Compile Data Set for Download or QSAR
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Found 10 Enz. Inhib. hit(s) with all data for entry = 50018913
LigandPNGBDBM50239948(CHEMBL4071326 | US9850225, Example 1166)
Affinity DataIC50:  3nMAssay Description:Inhibition of C-terminal his tagged human PD-1/human Fc tagged PDL-1 interaction expressed in HEK293 cells incubated for 2 hrs AlphaScreen assayMore data for this Ligand-Target Pair
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TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))TBA
LigandPNGBDBM50362641(CHEMBL384120)
Affinity DataIC50:  250nMAssay Description:Inhibition of his-tagged SARS-COV2 S-RBD binding to C-terminal Fc-tagged human ACE2 expressed in HEK293 cells incubated for 2 hrs by Alphascreen assa...More data for this Ligand-Target Pair
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TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))TBA
LigandPNGBDBM50613798(CHEMBL5267016)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of his-tagged SARS-COV2 S-RBD binding to C-terminal Fc-tagged human ACE2 expressed in HEK293 cells incubated for 2 hrs by Alphascreen assa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50613798(CHEMBL5267016)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of C-terminal his tagged human PD-1/human Fc tagged PDL-1 interaction expressed in HEK293 cells incubated for 2 hrs AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))TBA
LigandPNGBDBM50613799(CHEMBL5283695)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibition of his-tagged SARS-COV2 S-RBD binding to C-terminal Fc-tagged human ACE2 expressed in HEK293 cells incubated for 2 hrs by Alphascreen assa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50613799(CHEMBL5283695)
Affinity DataIC50:  3.70E+4nMAssay Description:Inhibition of C-terminal his tagged human PD-1/human Fc tagged PDL-1 interaction expressed in HEK293 cells incubated for 2 hrs AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50613800(CHEMBL5282197)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of C-terminal his tagged human PD-1/human Fc tagged PDL-1 interaction expressed in HEK293 cells incubated for 2 hrs AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))TBA
LigandPNGBDBM50613801(CHEMBL5276399)
Affinity DataIC50:  6.30E+4nMAssay Description:Inhibition of his-tagged SARS-COV2 S-RBD binding to C-terminal Fc-tagged human ACE2 expressed in HEK293 cells incubated for 2 hrs by Alphascreen assa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))TBA
LigandPNGBDBM50613800(CHEMBL5282197)
Affinity DataIC50:  6.50E+4nMAssay Description:Inhibition of his-tagged SARS-COV2 S-RBD binding to C-terminal Fc-tagged human ACE2 expressed in HEK293 cells incubated for 2 hrs by Alphascreen assa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50613801(CHEMBL5276399)
Affinity DataIC50:  6.60E+4nMAssay Description:Inhibition of C-terminal his tagged human PD-1/human Fc tagged PDL-1 interaction expressed in HEK293 cells incubated for 2 hrs AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed