Affinity DataKi: 1.10nMAssay Description:Antagonist at CCR5 (unknown origin) assessed as inhibitory constantMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Antagonist activity at CCR5 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 3.20nMAssay Description:Agonist activity at human N-terminal GLP-1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Agonist activity at PPARgamma (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Binding affinity to PPARgamma (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Antagonist activity at CCR2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 43nMAssay Description:Inverse agonist activity at LXRbeta in human HEK293 cells by luciferase reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 214nMAssay Description:Inverse agonist activity at LXRalpha in human HEK293 cells by luciferase reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 542nMAssay Description:Displacement of 125I-liraglutide from GLP-1 (unknown origin) by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.52E+7nMAssay Description:Agonist activity at PPARalpha (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 1nMAssay Description:Agonist activity at Gal4-fused PPARalpha LBD (unknown origin) transfected in human HepG2 cells assessed as transcriptional activation incubated for 2...More data for this Ligand-Target Pair
Affinity DataEC50: 100nMAssay Description:Agonist activity at PPARgamma (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Agonist activity at PPARdelta (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 175nMAssay Description:Agonist activity at PPARgamma (unknown origin) assessed as transcriptional activationMore data for this Ligand-Target Pair
Affinity DataEC50: 0.650nMAssay Description:Agonist activity at PPARalpha in human HepG2 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Agonist activity at PPARgamma in human HepG2 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 870nMAssay Description:Agonist activity at human PPARdeltaMore data for this Ligand-Target Pair
Affinity DataEC50: 210nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
Affinity DataEC50: 2.00E+4nMAssay Description:Binding affinity to PPARalpha (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 300nMAssay Description:Binding affinity to PPARgamma (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Agonist activity at PPARdelta (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 3.00E+4nMAssay Description:Agonist activity at PPARalpha (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 1.50E+3nMAssay Description:Agonist activity at human PPARalphaMore data for this Ligand-Target Pair
Affinity DataEC50: 5.00E+3nMAssay Description:Agonist activity at human PPARalphaMore data for this Ligand-Target Pair
Affinity DataEC50: 5.00E+7nMAssay Description:Agonist activity at mouse PPARalphaMore data for this Ligand-Target Pair
Affinity DataEC50: 5.50E+7nMAssay Description:Agonist activity at mouse PPARalphaMore data for this Ligand-Target Pair
Affinity DataEC50: 630nMAssay Description:Agonist activity at mouse PPARalphaMore data for this Ligand-Target Pair
Affinity DataEC50: 37nMAssay Description:Agonist activity at FXR (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 85nMAssay Description:Agonist activity at full length FXR in human Huh-7 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 99nMAssay Description:Agonist activity at FXR (unknown origin) by fluorescence resonance energy tranfer assayMore data for this Ligand-Target Pair
Affinity DataEC50: 45nMAssay Description:Agonist activity at PPARalpha (unknown origin) assessed as transcriptional activationMore data for this Ligand-Target Pair