TargetAdenosine receptor A1(Rattus norvegicus (rat))
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Binding affinity to adenosine A1 receptor in rat whole brain membranes by [3H]N6-cyclohexyladenosine displacement.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 2.40nMAssay Description:Binding affinity to adenosine A1 receptor in rat whole brain membranes by [3H]N6-cyclohexyladenosine displacement.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 4.60nMAssay Description:Binding affinity to adenosine A1 receptor in rat whole brain membranes by [3H]N6-cyclohexyladenosine displacement.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 6.80nMAssay Description:Binding affinity to adenosine A1 receptor in rat whole brain membranes by [3H]N6-cyclohexyladenosine displacement.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Binding affinity to adenosine A1 receptor in rat whole brain membranes by [3H]N6-cyclohexyladenosine displacement.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Binding affinity to adenosine A1 receptor in rat whole brain membranes by [3H]N6-cyclohexyladenosine displacement.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Binding affinity to adenosine A1 receptor in rat whole brain membranes by [3H]N6-cyclohexyladenosine displacement.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 23nMAssay Description:Binding affinity to adenosine A1 receptor in rat whole brain membranes by [3H]N6-cyclohexyladenosine displacement.More data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Binding affinity to A2 adenosine receptor in rat striatal membranes by [3H]NECA (1-(6-amino-9H-purin-9-yl)-1-deoxy-N-ethyl-beta-D-ribofuranuronamide)...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Binding affinity to A2 adenosine receptor in rat striatal membranes by [3H]NECA (1-(6-amino-9H-purin-9-yl)-1-deoxy-N-ethyl-beta-D-ribofuranuronamide)...More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:Binding affinity to adenosine A1 receptor in rat whole brain membranes by [3H]N6-cyclohexyladenosine displacement.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 49nMAssay Description:Binding affinity to adenosine A1 receptor in rat whole brain membranes by [3H]N6-cyclohexyladenosine displacement.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 79nMAssay Description:Binding affinity to adenosine A1 receptor in rat whole brain membranes by [3H]N6-cyclohexyladenosine displacement.More data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 98nMAssay Description:Binding affinity to A2 adenosine receptor in rat striatal membranes by [3H]NECA (1-(6-amino-9H-purin-9-yl)-1-deoxy-N-ethyl-beta-D-ribofuranuronamide)...More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 120nMAssay Description:Binding affinity to adenosine A1 receptor in rat whole brain membranes by [3H]N6-cyclohexyladenosine displacement.More data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 124nMAssay Description:Binding affinity to A2 adenosine receptor in rat striatal membranes by [3H]NECA (1-(6-amino-9H-purin-9-yl)-1-deoxy-N-ethyl-beta-D-ribofuranuronamide)...More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 146nMAssay Description:Binding affinity to adenosine A1 receptor in rat whole brain membranes by [3H]N6-cyclohexyladenosine displacement.More data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 161nMAssay Description:Binding affinity to A2 adenosine receptor in rat striatal membranes by [3H]NECA (1-(6-amino-9H-purin-9-yl)-1-deoxy-N-ethyl-beta-D-ribofuranuronamide)...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 280nMAssay Description:Binding affinity to A2 adenosine receptor in rat striatal membranes by [3H]NECA (1-(6-amino-9H-purin-9-yl)-1-deoxy-N-ethyl-beta-D-ribofuranuronamide)...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 290nMAssay Description:Binding affinity to A2 adenosine receptor in rat striatal membranes by [3H]NECA (1-(6-amino-9H-purin-9-yl)-1-deoxy-N-ethyl-beta-D-ribofuranuronamide)...More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 290nMAssay Description:Binding affinity to adenosine A1 receptor in rat whole brain membranes by [3H]N6-cyclohexyladenosine displacement.More data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 320nMAssay Description:Binding affinity to A2 adenosine receptor in rat striatal membranes by [3H]NECA (1-(6-amino-9H-purin-9-yl)-1-deoxy-N-ethyl-beta-D-ribofuranuronamide)...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 420nMAssay Description:Binding affinity to A2 adenosine receptor in rat striatal membranes by [3H]NECA (1-(6-amino-9H-purin-9-yl)-1-deoxy-N-ethyl-beta-D-ribofuranuronamide)...More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 480nMAssay Description:Binding affinity to adenosine A1 receptor in rat whole brain membranes by [3H]N6-cyclohexyladenosine displacement.More data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 660nMAssay Description:Binding affinity to A2 adenosine receptor in rat striatal membranes by [3H]NECA (1-(6-amino-9H-purin-9-yl)-1-deoxy-N-ethyl-beta-D-ribofuranuronamide)...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 1.23E+3nMAssay Description:Binding affinity to A2 adenosine receptor in rat striatal membranes by [3H]NECA (1-(6-amino-9H-purin-9-yl)-1-deoxy-N-ethyl-beta-D-ribofuranuronamide)...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 1.72E+3nMAssay Description:Binding affinity to A2 adenosine receptor in rat striatal membranes by [3H]NECA (1-(6-amino-9H-purin-9-yl)-1-deoxy-N-ethyl-beta-D-ribofuranuronamide)...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 2.20E+3nMAssay Description:Binding affinity to A2 adenosine receptor in rat striatal membranes by [3H]NECA (1-(6-amino-9H-purin-9-yl)-1-deoxy-N-ethyl-beta-D-ribofuranuronamide)...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 3.80E+3nMAssay Description:Binding affinity to A2 adenosine receptor in rat striatal membranes by [3H]NECA (1-(6-amino-9H-purin-9-yl)-1-deoxy-N-ethyl-beta-D-ribofuranuronamide)...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 4.70E+3nMAssay Description:Binding affinity to A2 adenosine receptor in rat striatal membranes by [3H]NECA (1-(6-amino-9H-purin-9-yl)-1-deoxy-N-ethyl-beta-D-ribofuranuronamide)...More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 1.43E+4nMAssay Description:Binding affinity to adenosine A1 receptor in rat whole brain membranes by [3H]N6-cyclohexyladenosine displacement.More data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Parke-Davis Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 2.60E+4nMAssay Description:Binding affinity to A2 adenosine receptor in rat striatal membranes by [3H]NECA (1-(6-amino-9H-purin-9-yl)-1-deoxy-N-ethyl-beta-D-ribofuranuronamide)...More data for this Ligand-Target Pair