Affinity DataKi: 110nMAssay Description:Binding of Adenosine A2 receptor in whole rat brain membrane using [3H]CHA as a RadioligandMore data for this Ligand-Target Pair
Affinity DataKi: 660nMAssay Description:Binding affinity to A2 adenosine receptor in rat striatal membranes by [3H]NECA (1-(6-amino-9H-purin-9-yl)-1-deoxy-N-ethyl-beta-D-ribofuranuronamide)...More data for this Ligand-Target Pair
Affinity DataKi: 663nMAssay Description:Affinity for adenosine A2 receptor at rat striatal membrane using 5 nM [3H]CGS-21680More data for this Ligand-Target Pair
Affinity DataKi: 1.20E+3nMAssay Description:Inhibition of [3H]- NECA binding to adenosine receptor A2More data for this Ligand-Target Pair
Affinity DataKi: 5.00E+4nMAssay Description:Binding affinity for Adenosine A2 receptor in corpora striata of rats using [3H]NECAMore data for this Ligand-Target Pair
Affinity DataIC50: 660nMAssay Description:Displacement of [3H]-NECA from adenosine A2 receptor of rat striatal membraneMore data for this Ligand-Target Pair