TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataKi: 0.400nMAssay Description:Binding affinity to CXCR3More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:Binding affinity to AT1 receptorMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:Binding affinity to AT1 receptorMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Binding affinity to ETA receptorMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Binding affinity to CCR1More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Antagonist activity at human CCR3 assessed as inhibition of CCL11-induced calcium influx by cell based assayMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataKi: 2.30nMAssay Description:Binding affinity to CCR1More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataKi: 9.30nMAssay Description:Binding affinity to ETA receptorMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Binding affinity to CCR4More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity to histamine H1 receptorMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Binding affinity to TXA2 receptor receptorMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity to histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Antagonist activity at histamine H1 receptor expressed in human PC3 cells inhibition of histamine-induced calcium influx by cell based assayMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataKi: 66nMAssay Description:Binding affinity to CCR5More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataKi: 74nMAssay Description:Binding affinity to CCR1More data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataKi: 740nMAssay Description:Binding affinity to TXA2 receptor receptorMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to TXA2 receptor receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataKi: 1.32E+3nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to AT1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+4nMAssay Description:Binding affinity to ETA receptorMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataIC50: 0.0340nMAssay Description:Antagonist activity at CCR3 assessed as inhibition of chemotaxis by cell based assayMore data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataIC50: 0.0490nMAssay Description:Binding affinity to CXCR2More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataIC50: 0.170nMAssay Description:Binding affinity to CCR5More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataIC50: 0.320nMAssay Description:Binding affinity to CCR5More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataIC50: 0.450nMAssay Description:Binding affinity to CCR5More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Antagonist activity at CXCR2 assessed as inhibition of CXCL8-induced neutrophil chemotaxisMore data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Binding affinity to CXCR1More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataIC50: 1.40nMAssay Description:Binding affinity to CCR5More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Binding affinity to CCR3More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 9(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataIC50: 2.80nMAssay Description:Antagonist activity at CCR9 assessed as inhibition of CCL25-induced chemotaxis by cell based assayMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Antagonist activity at CCR5 assessed as inhibition of CCL3 bindingMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Binding affinity to CCR5More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataIC50: 3.10nMAssay Description:Binding affinity to CCR5More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataIC50: 3.40nMAssay Description:Antagonist activity at CCR1 assessed as inhibition of CCL3-induced chemotaxis by cell based assayMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataIC50: 3.60nMAssay Description:Binding affinity to CCR2More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataIC50: 3.90nMAssay Description:Binding affinity to CXCR1More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Binding affinity to CCR2More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Antagonist activity at CCR1More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataIC50: 5.10nMAssay Description:Binding affinity to CXCR2More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataIC50: 5.90nMAssay Description:Antagonist activity at CCR2 assessed as inhibition of CCL2 bindingMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 9(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Binding affinity to CCR9More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Binding affinity to CXCR3More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataIC50: 8.10nMAssay Description:Antagonist activity at CCR3 assessed as inhibition of eotaxin bindingMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataIC50: 9.60nMAssay Description:Antagonist activity at CCR1 assessed as inhibition of CCL3-induced chemotaxis by cell based assayMore data for this Ligand-Target Pair