Affinity DataIC50: 0.5nMAssay Description:Antagonist activity at human adenosine 2A receptor expressed in HEK293 cells assessed as reduction in cAMP production preincubated for 10 mins follow...More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Antagonist activity at human adenosine 2A receptor expressed in HEK293 cells assessed as reduction in cAMP production preincubated for 10 mins follow...More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Antagonist activity at adenosine 2A receptor in human peripheral blood lymphocytes assessed as reduction in NECA-stimulated CREB phosphorylation by f...More data for this Ligand-Target Pair
Affinity DataIC50: 49nMAssay Description:Antagonist activity at human adenosine 2A receptor expressed in HEK293 cells assessed as reduction in cAMP production preincubated for 10 mins follow...More data for this Ligand-Target Pair