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Compile Data Set for Download or QSAR
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Found
1
Enz. Inhib. hit(s) with Target = 'Glutaminase kidney isoform, mitochondrial [63-669]' and Ligand = 'BDBM387007'
Target
Glutaminase kidney isoform, mitochondrial [63-669]
(Homo sapiens (Human))
Astrazeneca
US Patent
Ligand
BDBM387007
((2S)-N-[5-[[(3R)-1-(6-Fluoropyridazin-3-yl)pyrroli...)
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Affinity Data
IC50: 30.3nM
Assay Description:
A Glutamate Oxidase/AmplexRed coupled assay was used to measure the ability of compounds to bind to and inhibit the activity of GLS1 in vitro. 6His t...
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Target Info
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Ligand Info
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US Patent
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