Found 4 Enz. Inhib. hit(s) with Target = 'Metabotropic glutamate receptor 4' and Ligand = 'BDBM50255292'
Affinity DataEC50: 160nMAssay Description:Agonist activity at mGlu4 (unknown origin) expressed in HEK293 cells coexpressing chimeric Gq/i protein assessed as [3H]inositol phosphate accumulati...More data for this Ligand-Target Pair
Affinity DataEC50: 190nMAssay Description:Agonist activity at mGlu4 (unknown origin) expressed in HEK293 cells coexpressing chimeric Gq/i protein assessed as [3H]inositol phosphate accumulati...More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataEC50: 9.32E+3nMAssay Description:Agonist activity at mGlu4 (unknown origin) expressed in HEK293 cells coexpressing chimeric Gq/i protein assessed as [3H]inositol phosphate accumulati...More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
University of Paris
Curated by ChEMBL
University of Paris
Curated by ChEMBL
Affinity DataEC50: 320nMAssay Description:Agonist activity at mGlu4 in Wistar rat striatum assessed as decrease in striatal GABAergic inhibitory post-synaptic potential by whole cell patch cl...More data for this Ligand-Target Pair