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Found 4 Enz. Inhib. hit(s) with Target = 'O-acetylserine sulfhydrylase' and Ligand = 'BDBM50427257'
TargetO-acetylserine sulfhydrylase(Mycobacterium tuberculosis)
Karolinska Institutet

Curated by ChEMBL
LigandPNGBDBM50427257(CHEMBL2325118)
Affinity DataKi:  5.00E+3nMAssay Description:Competitive inhibition of Mycobacterium tuberculosis CysK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetO-acetylserine sulfhydrylase(Mycobacterium tuberculosis)
Karolinska Institutet

Curated by ChEMBL
LigandPNGBDBM50427257(CHEMBL2325118)
Affinity DataKi:  5.00E+3nMAssay Description:Competitive inhibition of Mycobacterium tuberculosis CysK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetO-acetylserine sulfhydrylase(Mycobacterium tuberculosis)
Karolinska Institutet

Curated by ChEMBL
LigandPNGBDBM50427257(CHEMBL2325118)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis CysK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetO-acetylserine sulfhydrylase(Mycobacterium tuberculosis)
Karolinska Institutet

Curated by ChEMBL
LigandPNGBDBM50427257(CHEMBL2325118)
Affinity DataIC50:  7.40E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis CysK1 using O-acetyl-L-serine as substrate assessed as L-cycteine formation after 5 mins by spectrophotometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed