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Found 3 Enz. Inhib. hit(s) with Target = 'Potassium voltage-gated channel subfamily KQT member 2/3' and Ligand = 'BDBM50595542'
TargetPotassium voltage-gated channel subfamily KQT member 2/3(Homo sapiens (Human))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM50595542(CHEMBL5204124)
Affinity DataEC50:  3.20E+3nMAssay Description:Activation of Kv7.2/Kv7.3 channel (unknown origin) expressed in CHO cells assessed as slope of fluorescent signal by FluxOR fluorescent dye based ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2/3(Homo sapiens (Human))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM50595542(CHEMBL5204124)
Affinity DataEC50:  60nMAssay Description:Activation of Kv7.2/Kv7.3 channel (unknown origin) expressed in CHO cells assessed as maximum current density measured after 24 hrs by whole cell pat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2/3(Homo sapiens (Human))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM50595542(CHEMBL5204124)
Affinity DataEC50:  150nMAssay Description:Activation of Kv7.2/Kv7.3 channel (unknown origin) expressed in CHO cells at + 80 mV assessed as leftward shift change in half activation potential m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed