Report error Found 4 Enz. Inhib. hit(s) with Target = 'Proprotein convertase subtilisin/kexin type 9' and Ligand = 'BDBM50609098'
TargetProprotein convertase subtilisin/kexin type 9(Human)
Aligarh Muslim University
Curated by ChEMBL
Aligarh Muslim University
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of human PCSK9 preincubated for 30 mins followed by ab20 addition and measured after 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
TargetProprotein convertase subtilisin/kexin type 9(Human)
Aligarh Muslim University
Curated by ChEMBL
Aligarh Muslim University
Curated by ChEMBL
Affinity DataIC50: 720nMAssay Description:Inhibition of human PCSK9 preincubated for 30 mins followed by EGF(A) addition and measured after 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
TargetProprotein convertase subtilisin/kexin type 9(Human)
Aligarh Muslim University
Curated by ChEMBL
Aligarh Muslim University
Curated by ChEMBL
Affinity DataIC50: 1.83E+3nMAssay Description:Inhibition of human PCSK9 preincubated for 30 mins followed by LDLR addition and measured after 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
TargetProprotein convertase subtilisin/kexin type 9(Human)
Aligarh Muslim University
Curated by ChEMBL
Aligarh Muslim University
Curated by ChEMBL
Affinity DataKd: 390nMAssay Description:Binding affinity to human PCSK9More data for this Ligand-Target Pair