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Compile Data Set for Download or QSAR
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Found
1
Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase JAK2' and Ligand = 'BDBM212271'
Target
Tyrosine-protein kinase JAK2
(Homo sapiens (Human))
Gilead Sciences
Curated by
ChEMBL
Ligand
BDBM212271
(6-(6-aminopyrazin-2-yl)-N-(4-(4-(oxetan-3-yl)piper...)
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Affinity Data
IC50: 120nM
Assay Description:
Inhibition of wild-type human partial length JAK2 JH1 catalytic domain (A829 to G1132 residues) expressed in mammalian expression system by Kinomesca...
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Target Info
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