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Found 1 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase JAK2' and Ligand = 'BDBM212271'
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM212271(6-(6-aminopyrazin-2-yl)-N-(4-(4-(oxetan-3-yl)piper...)
Affinity DataIC50:  120nMAssay Description:Inhibition of wild-type human partial length JAK2 JH1 catalytic domain (A829 to G1132 residues) expressed in mammalian expression system by Kinomesca...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed