Affinity DataKi: 0.910nMAssay Description:Binding affinity towards opioid Delta receptor using [3H]DADLE as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.910nMAssay Description:Binding affinity towards opioid Delta receptor using [3H]DADLE as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinity towards opioid Delta receptor using [3H]DADLE as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinity towards opioid Delta receptor using [3H]DADLE as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 5.60nMAssay Description:Binding affinity towards opioid Delta receptor using [3H]DADLE as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity towards opioid Delta receptor using [3H]DADLE as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity towards opioid Delta receptor using [3H]DADLE as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Binding affinity towards opioid Mu receptor using [3H]DAMGO as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Binding affinity towards opioid Mu receptor using [3H]DAMGO as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Binding affinity towards opioid Delta receptor using [3H]DADLE as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 139nMAssay Description:Binding affinity towards opioid Delta receptor using [3H]DADLE as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.21E+3nMAssay Description:Binding affinity towards opioid Mu receptor using [3H]DAMGO as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.21E+3nMAssay Description:Binding affinity towards opioid Mu receptor using [3H]DAMGO as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.45E+3nMAssay Description:Binding affinity towards opioid kappa receptor using [3H]U-69593 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.59E+3nMAssay Description:Binding affinity towards opioid Mu receptor using [3H]DAMGO as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.61E+3nMAssay Description:Binding affinity towards opioid Mu receptor using [3H]DAMGO as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.61E+3nMAssay Description:Binding affinity towards opioid Mu receptor using [3H]DAMGO as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2.62E+3nMAssay Description:Binding affinity towards opioid Mu receptor using [3H]DAMGO as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3.28E+3nMAssay Description:Binding affinity towards opioid kappa receptor using [3H]U-69593 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3.28E+3nMAssay Description:Binding affinity towards opioid kappa receptor using [3H]U-69593 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3.54E+3nMAssay Description:Binding affinity towards opioid kappa receptor using [3H]U-69593 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3.54E+3nMAssay Description:Binding affinity towards opioid kappa receptor using [3H]U-69593 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3.72E+3nMAssay Description:Binding affinity towards opioid kappa receptor using [3H]U-69593 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 8.70E+3nMAssay Description:Binding affinity towards opioid kappa receptor using [3H]U-69593 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards opioid Mu receptor using [3H]DAMGO as radioligandMore data for this Ligand-Target Pair
Affinity DataKd: 684nMAssay Description:Binding affinity against Mu opioid receptor using [35S]GTP-gamma-S, binding assay in guinea pig caudate membranes in unblocked conditionMore data for this Ligand-Target Pair
Affinity DataKd: 4.67E+3nMAssay Description:Binding affinity against Delta opioid receptor in using [35S]GTP-gamma-S, binding assay in guinea pig caudate membranes blocked with 20 nM NTIMore data for this Ligand-Target Pair
Affinity DataKd: 673nMAssay Description:Binding affinity against Mu opioid receptor using [35S]GTP-gamma-S, binding assay in guinea pig caudate membranes blocked with 6000 nM CTAPMore data for this Ligand-Target Pair
Affinity DataKd: 2.14E+3nMAssay Description:Binding affinity against Mu opioid receptor using [35S]GTP-gamma-S, binding assay in guinea pig caudate membranes blocked with 6000 nM CTAPMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKd: 4.89E+3nMAssay Description:Binding affinity against Mu opioid receptor using [35S]GTP-gamma-S, binding assay in guinea pig caudate membranes blocked with 6000 nM CTAPMore data for this Ligand-Target Pair
Affinity DataKd: 1.98E+3nMAssay Description:Binding affinity against kappa opioid receptor using [35S]GTP-gamma-S, binding assay in guinea pig caudate membranes blocked with 6 nM nor-BNIMore data for this Ligand-Target Pair
Affinity DataKd: 317nMAssay Description:Binding affinity against kappa opioid receptor using [35S]GTP-gamma-S, binding assay in guinea pig caudate membranes blocked with 6 nM nor-BNIMore data for this Ligand-Target Pair
Affinity DataKd: 2.14E+3nMAssay Description:Binding affinity against Mu opioid receptor using [35S]GTP-gamma-S, binding assay in guinea pig caudate membranes blocked with 6000 nM CTAPMore data for this Ligand-Target Pair
Affinity DataKd: 3.50E+3nMAssay Description:Binding affinity against Mu opioid receptor using [35S]GTP-gamma-S, binding assay in guinea pig caudate membranes in unblocked conditionMore data for this Ligand-Target Pair
Affinity DataKd: 1.98E+3nMAssay Description:Binding affinity against Mu opioid receptor using [35S]GTP-gamma-S, binding assay in guinea pig caudate membranes in unblocked conditionMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKd: 4.89E+3nMAssay Description:Binding affinity against Delta opioid receptor in using [35S]GTP-gamma-S, binding assay in guinea pig caudate membranes blocked with 20 nM NTIMore data for this Ligand-Target Pair
Affinity DataKd: 684nMAssay Description:Binding affinity against Mu opioid receptor using [35S]GTP-gamma-S, binding assay in guinea pig caudate membranes in unblocked conditionMore data for this Ligand-Target Pair
Affinity DataKd: 577nMAssay Description:Binding affinity against Mu opioid receptor using [35S]GTP-gamma-S, binding assay in guinea pig caudate membranes in unblocked conditionMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKd: 2.95E+3nMAssay Description:Binding affinity against kappa opioid receptor using [35S]GTP-gamma-S, binding assay in guinea pig caudate membranes blocked with 6 nM nor-BNIMore data for this Ligand-Target Pair
Affinity DataKd: 629nMAssay Description:Binding affinity against kappa opioid receptor using [35S]GTP-gamma-S, binding assay in guinea pig caudate membranes blocked with 6 nM nor-BNIMore data for this Ligand-Target Pair
Affinity DataKd: 1.85E+3nMAssay Description:Binding affinity against Delta opioid receptor in using [35S]GTP-gamma-S, binding assay in guinea pig caudate membranes blocked with 20 nM NTIMore data for this Ligand-Target Pair
Affinity DataKd: 592nMAssay Description:Binding affinity against Mu opioid receptor using [35S]GTP-gamma-S, binding assay in guinea pig caudate membranesin unblocked conditionMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKd: 509nMAssay Description:Binding affinity against kappa opioid receptor using [35S]GTP-gamma-S, binding assay in guinea pig caudate membranes blocked with 6 nM nor-BNIMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKd: 3.72E+3nMAssay Description:Binding affinity against kappa opioid receptor using [35S]GTP-gamma-S, binding assay in guinea pig caudate membranes blocked with 6 nM nor-BNIMore data for this Ligand-Target Pair
Affinity DataKd: 3.60E+3nMAssay Description:Binding affinity against Mu opioid receptor using [35S]GTP-gamma-S, binding assay in guinea pig caudate membranes blocked with 6000 nM CTAPMore data for this Ligand-Target Pair
Affinity DataKd: 3.50E+3nMAssay Description:Binding affinity against Mu opioid receptor using [35S]GTP-gamma-S, binding assay in guinea pig caudate membranes in unblocked conditionMore data for this Ligand-Target Pair
Affinity DataKd: 317nMAssay Description:Binding affinity against Mu opioid receptor using [35S]GTP-gamma-S, binding assay in guinea pig caudate membranes in unblocked conditionMore data for this Ligand-Target Pair
Affinity DataKd: 592nMAssay Description:Binding affinity against Mu opioid receptor using [35S]GTP-gamma-S, binding assay in guinea pig caudate membranesin unblocked conditionMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKd: 3.72E+3nMAssay Description:Binding affinity against kappa opioid receptor using [35S]GTP-gamma-S, binding assay in guinea pig caudate membranes blocked with 6 nM nor-BNIMore data for this Ligand-Target Pair
Affinity DataKd: 4.67E+3nMAssay Description:Binding affinity against Mu opioid receptor using [35S]GTP-gamma-S, binding assay in guinea pig caudate membranes blocked with 6000 nM CTAPMore data for this Ligand-Target Pair