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TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50590650(CHEMBL5204619)
Affinity DataKi:  0.5nMAssay Description:Binding affinity to cerebrum 5-HT2 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50007551(Enantiomer 1'3'-chlorospiro[2-cyclohexene-1,5'-(10...)
Affinity DataKi:  0.570nMAssay Description:The compound was tested for binding affinity against 5-hydroxytryptamine 2 receptor using ketanserin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50007551(Enantiomer 1'3'-chlorospiro[2-cyclohexene-1,5'-(10...)
Affinity DataKi:  0.570nMAssay Description:The compound was tested for binding affinity against 5-hydroxytryptamine 2 receptor using ketanserin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50007550(3'-chlorospiro[2-cyclohexene-1,5'-(10',11'-dihydro...)
Affinity DataKi:  1nMAssay Description:The compound was tested for binding affinity against 5-hydroxytryptamine 2 receptor using ketanserin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50007550(3'-chlorospiro[2-cyclohexene-1,5'-(10',11'-dihydro...)
Affinity DataKi:  1nMAssay Description:The compound was tested for binding affinity against 5-hydroxytryptamine 2 receptor using ketanserin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50001884(8-Chloro-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b...)
Affinity DataKi:  5nMAssay Description:In vitro binding affinity for 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2018
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM35254(CHEMBL715 | 2-methyl-4-(4-methylpiperazin-1-yl)-10...)
Affinity DataKi:  10nMAssay Description:In vitro binding affinity of compound against neuronal 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50130272(2a-[3-(4-Phenyl-piperazin-1-yl)-propyl]-2a,3,4,5-t...)
Affinity DataKi:  16nMAssay Description:Binding affinity towards 5-HT2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50289291([10-(4-Methyl-piperazin-1-yl)-4H-3-thia-4,9-diaza-...)
Affinity DataKi:  18nMAssay Description:In vitro binding affinity of compound against neuronal 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  20nMAssay Description:In vitro binding affinity for 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2018
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50283335(1-Phenethyl-4-[2-(3-phenyl-prop-2-ynyloxy)-ethyl]-...)
Affinity DataKi:  21nMAssay Description:Binding affinity towards 5-HT2 receptor using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50240701(CHEMBL1125 | 2-Methyl-10-piperazin-1-yl-4H-3-thia-...)
Affinity DataKi:  23nMAssay Description:In vitro binding affinity of compound against neuronal 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50001115(CHEMBL103983 | 8-[(3-Phenyl-propylamino)-methyl]-7...)
Affinity DataKi:  28nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptor expressed in CHO cell membranes using [3H]ketanserin (60 Ci/mmol, 1 nM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50283326(1-Benzyl-4-(3,3-diphenyl-allyloxymethyl)-piperidin...)
Affinity DataKi:  29nMAssay Description:Binding affinity towards 5-HT2 receptor using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50283331(1-Benzyl-4-[(E)-3-(4-fluoro-phenyl)-allyloxymethyl...)
Affinity DataKi:  31nMAssay Description:Binding affinity towards 5-HT2 receptor using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50218629(CHEMBL282927)
Affinity DataKi:  32nMAssay Description:In vitro binding affinity for 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2018
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50001116(CHEMBL418802 | 8-[4-(2-Oxo-2,3-dihydro-benzoimidaz...)
Affinity DataKi:  32nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptor expressed in CHO cell membranes using [3H]ketanserin (60 Ci/mmol, 1 nM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50088844(4-{4-[4-(4-Phenyl-piperazin-1-yl)-butyl]-phenyl}-t...)
Affinity DataKi:  37nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50001117(CHEMBL318374 | 8-[(3-Phenyl-propylamino)-methyl]-7...)
Affinity DataKi:  39nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptor expressed in CHO cell membranes using [3H]ketanserin (60 Ci/mmol, 1 nM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50283322(1-Benzyl-4-((E)-3-phenyl-allyloxymethyl)-piperidin...)
Affinity DataKi:  44nMAssay Description:Binding affinity towards 5-HT2 receptor using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50088839(N-{4-[4-(4-Phenyl-piperazin-1-yl)-butyl]-benzyl}-a...)
Affinity DataKi:  48nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50133917(((6S,7R)-6-Methyl-6,7,8,9-tetrahydro-naphtho[1,2-b...)
Affinity DataKi:  70nMAssay Description:Tested in vitro for the inhibition of [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor, expressed in cloned CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50283320(1-Phenethyl-4-(3-phenyl-prop-2-ynyloxy)-piperidine...)
Affinity DataKi:  72nMAssay Description:Binding affinity towards 5-HT2 receptor using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50283336(4-{2-[3-(4-Fluoro-phenyl)-prop-2-ynyloxy]-ethyl}-1...)
Affinity DataKi:  81nMAssay Description:Binding affinity towards 5-HT2 receptor using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50283321(1-[2-(4-Fluoro-phenyl)-ethyl]-4-[2-(3-phenyl-prop-...)
Affinity DataKi:  85nMAssay Description:Binding affinity towards 5-HT2 receptor using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50001109(CHEMBL102175 | 8-(4-Oxo-1-phenyl-1,3,8-triaza-spir...)
Affinity DataKi:  93nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptor expressed in CHO cell membranes using [3H]ketanserin (60 Ci/mmol, 1 nM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50116963(2a-[4-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-butyl...)
Affinity DataKi:  98nMAssay Description:Binding affinity towards 5-HT2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50283394((E)-N-(1-Benzyl-piperidin-4-yl)-3-phenyl-acrylamid...)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50289292(2-Methyl-10-(4-methyl-4-oxy-piperazin-1-yl)-4H-3-t...)
Affinity DataKi:  112nMAssay Description:In vitro binding affinity of compound against neuronal 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50088846(N-{4-[2-(4-Phenyl-piperazin-1-yl)-ethyl]-benzyl}-a...)
Affinity DataKi:  130nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50001110(CHEMBL318166 | 8-(4-Oxo-1-phenyl-1,3,8-triaza-spir...)
Affinity DataKi:  143nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptor expressed in CHO cell membranes using [3H]ketanserin (60 Ci/mmol, 1 nM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50290663((7aR,10aS)-8-Propyl-7,7a,8,9,10,10a-hexahydro-6H-1...)
Affinity DataKi:  146nMAssay Description:Tested in vitro for the inhibition of [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor, expressed in cloned CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50088841(N-{4-[3-(4-Phenyl-piperazin-1-yl)-propyl]-benzyl}-...)
Affinity DataKi:  160nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50001111(CHEMBL319023 | 8-(4-Ethoxycarbonyl-piperidin-1-ylm...)
Affinity DataKi:  170nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptor expressed in CHO cell membranes using [3H]ketanserin (60 Ci/mmol, 1 nM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50001120(CHEMBL101483 | 8-(4-Carbamoyl-4-phenylamino-piperi...)
Affinity DataKi:  171nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptor expressed in CHO cell membranes using [3H]ketanserin (60 Ci/mmol, 1 nM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50002268(CHEMBL337810 | CHEMBL80656 | 1-Benzyl-4-(3-phenyl-...)
Affinity DataKi:  180nMAssay Description:Binding affinity towards 5-HT2 receptor using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50095890(2-[2-(4-dibenzo[b,f][1,4]thiazepin-11-ylpiperazin-...)
Affinity DataKi:  220nMAssay Description:In vitro binding affinity for 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2018
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50283328(1-Phenethyl-4-((E)-3-phenyl-allyloxymethyl)-piperi...)
Affinity DataKi:  250nMAssay Description:Binding affinity towards 5-HT2 receptor using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50283329(1-Benzyl-4-(3-phenyl-prop-2-ynyloxymethyl)-piperid...)
Affinity DataKi:  254nMAssay Description:Binding affinity towards 5-HT2 receptor using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50283404((1-Benzyl-piperidin-4-yl)-phenyl-(3-phenyl-prop-2-...)
Affinity DataKi:  280nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50283393(3-Phenyl-propynoic acid (1-benzyl-piperidin-4-yl)-...)
Affinity DataKi:  280nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50001119(CHEMBL101535 | 8-(4-Oxo-1-phenyl-1,3,8-triaza-spir...)
Affinity DataKi:  281nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptor expressed in CHO cell membranes using [3H]ketanserin (60 Ci/mmol, 1 nM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50283333(4-((E)-3-Phenyl-allyloxymethyl)-1-(3-phenyl-propyl...)
Affinity DataKi:  283nMAssay Description:Binding affinity towards 5-HT2 receptor using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50283324(1-Naphthalen-1-ylmethyl-4-((E)-3-phenyl-allyloxyme...)
Affinity DataKi:  284nMAssay Description:Binding affinity towards 5-HT2 receptor using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50283405((1-Benzyl-piperidin-4-yl)-methyl-(3-phenyl-prop-2-...)
Affinity DataKi:  320nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50283325(1-Benzyl-4-[(E)-3-(4-trifluoromethyl-phenyl)-allyl...)
Affinity DataKi:  324nMAssay Description:Binding affinity towards 5-HT2 receptor using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50283337(1-Benzyl-4-((1E,3E)-4-phenyl-buta-1,3-dienyloxymet...)
Affinity DataKi:  547nMAssay Description:Binding affinity towards 5-HT2 receptor using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50283396((1-Benzyl-piperidin-4-yl)-bis-((E)-3-phenyl-allyl)...)
Affinity DataKi:  550nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50283330(1-((E)-But-2-enyl)-4-((E)-3-phenyl-allyloxymethyl)...)
Affinity DataKi:  650nMAssay Description:Binding affinity towards 5-HT2 receptor using [3H]ketanserin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetSerotonin 2 (5-HT2) receptor(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50283400((1-Benzyl-piperidin-4-yl)-methyl-((E)-3-phenyl-all...)
Affinity DataKi:  840nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

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