Compile Data Set for Download or QSAR
maximum 50k data
Found 4 of ic50 for monomerid = 119763
TargetMelanin-concentrating hormone receptor 1(Mus musculus)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM119763(US8685958, 12)
Affinity DataIC50:  15nMAssay Description:Displacement of [125I]Tyr13-MCH from mouse MCHR1 after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM119763(US8685958, 12)
Affinity DataIC50:  45nMAssay Description:Melanin Concentrating Hormone Receptor 1 (MCHR1) is a G-protein coupled receptor that interacts with heterotrimeric G proteins containing a Gαi/...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Astrazeneca

US Patent
LigandPNGBDBM119763(US8685958, 12)
Affinity DataIC50:  45nMAssay Description:Antagonist activity at human MCHR1 expressed in CHO cell membranes preincubated for 5 mins followed by addition of MCH peptide measured after 45 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM119763(US8685958, 12)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of human ERG by IonWork assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed