Compile Data Set for Download or QSAR
maximum 50k data
Found 5 of ic50 for monomerid = 50065210
LigandPNGBDBM50065210(1-Aza-bicyclo[2.2.1]heptan-3-one O-nona-2,5,8-triy...)
Affinity DataIC50:  8nMAssay Description:Effective concentration for HMPA (human muscarinic inositol phosphate accumulation) activity measured in CHO cells expressing Muscarinic acetylcholin...More data for this Ligand-Target Pair
In DepthDetails Article
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50065210(1-Aza-bicyclo[2.2.1]heptan-3-one O-nona-2,5,8-triy...)
Affinity DataIC50:  2.03E+3nMAssay Description:Inhibitory activity against human Muscarinic acetylcholine receptor M1 using [3H]-quinuclidinyl benzilate to label antagonist site (RQNB) in CHO cell...More data for this Ligand-Target Pair
In DepthDetails Article
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50065210(1-Aza-bicyclo[2.2.1]heptan-3-one O-nona-2,5,8-triy...)
Affinity DataIC50:  2.03E+3nMAssay Description:Binding affinity of [3H]-QNB to CHO cells expressing human Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50065210(1-Aza-bicyclo[2.2.1]heptan-3-one O-nona-2,5,8-triy...)
Affinity DataIC50:  2.18E+3nMAssay Description:Inhibitory activity against human Muscarinic acetylcholine receptor M2 using [3H]-quinuclidinyl benzilate to label antagonist site (RQNB) in CHO cell...More data for this Ligand-Target Pair
In DepthDetails Article
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50065210(1-Aza-bicyclo[2.2.1]heptan-3-one O-nona-2,5,8-triy...)
Affinity DataIC50:  2.18E+3nMAssay Description:Binding affinity of [3H]-QNB to CHO cells expressing human Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed