Affinity DataIC50: 56.6nMAssay Description:Displacement of [3H]DAMGO from Wistar rat mu opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of North Carolina At Wilmington
Curated by ChEMBL
University Of North Carolina At Wilmington
Curated by ChEMBL
Affinity DataIC50: 320nMAssay Description:Inhibitory activity against non-selective opiate receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 552nMAssay Description:In vitro inhibitory activity against mu opioid receptor using guinea pig ileum (GPI) assayMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Medical University Of Lodz
Curated by ChEMBL
Medical University Of Lodz
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H][Ile5,6]deltorphin 2 from delta opioid receptor in Wistar rat brain membrane by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 3.69E+3nMAssay Description:In vitro inhibitory activity against delta opioid receptor using mouse vas deferens (MVD) assayMore data for this Ligand-Target Pair