Compile Data Set for Download or QSAR
maximum 50k data
Found 4 of ki for monomerid = 50407330
TargetMuscarinic acetylcholine receptor M2(RAT)
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50407330(CHEMBL2112939)
Affinity DataKi:  2.20nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M2 was determined by measuring its ability to displace [3H]-AF-DX 384 from rat he...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic receptor M1(Bos taurus)
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50407330(CHEMBL2112939)
Affinity DataKi:  7.40nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M1 was determined by measuring its ability to displace [3H]-Pirenzepine from bovi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50407330(CHEMBL2112939)
Affinity DataKi:  62.1nMAssay Description:In vitro binding affinity towards Sigma receptor type 1 was determined by measuring its ability to displace [3H]-(+)-pentazocine from guinea pig brai...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50407330(CHEMBL2112939)
Affinity DataKi:  80nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M3 was determined by measuring its ability to displace [3H]-N-methyl- scopolamine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed