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Found 2 Enz. Inhib. hit(s) with Target = '1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial' and Ligand = 'BDBM50155472'
Target1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial(Rattus norvegicus)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50155472(6-Methoxy-2-[1-o-tolyl-meth-(E)-ylidene]-3,4-dihyd...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibitory activity against 25-hydroxyvitamin D3 24-hydroxylase of rat kidney mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial(Homo sapiens (Human))
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50155472(6-Methoxy-2-[1-o-tolyl-meth-(E)-ylidene]-3,4-dihyd...)
Affinity DataIC50:  4.80E+5nMAssay Description:Inhibition of CYP24A1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed