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Found 1 Enz. Inhib. hit(s) with Target = '11-beta-hydroxysteroid dehydrogenase type 2' and Ligand = 'BDBM50339809'
Target11-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
University Of Technology

Curated by ChEMBL
LigandPNGBDBM50339809((5aR,7aR,7bS,9aS,12S,13aR,15aR,15bS)-2,3,4,5,5a,6,...)
Affinity DataIC50:  11nMAssay Description:Inhibition of human 11beta-HSD2 expressed in HEK293 cells assessed as conversion of [1,2,6,7-[3H]cortisol to cortisone after 10 mins by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed