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Found 2 Enz. Inhib. hit(s) with Target = '17-beta-hydroxysteroid dehydrogenase type 1' and Ligand = 'BDBM50232146'
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Pharmbiotec

Curated by ChEMBL
LigandPNGBDBM50232146(CHEMBL4092593)
Affinity DataIC50:  7nMAssay Description:Inhibition of human placental cytosolic 17beta-HSD1 using [3H]-E1 as substrate after 10 mins in presence of NADPH by radio-flow detector based analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 1(Homo sapiens (Human))
Pharmbiotec

Curated by ChEMBL
LigandPNGBDBM50232146(CHEMBL4092593)
Affinity DataIC50:  7.20nMAssay Description:Inhibition of human placental cytosolic 17beta-HSD1 assessed as reduction in activation of [2,4,6,7-3H]-E1 substrate to E2 after 10 mins in presence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed