Compile Data Set for Download or QSAR
Report error Found 1 Enz. Inhib. hit(s) with Target = '3-phosphoinositide-dependent protein kinase 1 [51-359,A162V]' and Ligand = 'BDBM17055'
LigandPNGBDBM17055((9S)-9-[(dimethylamino)methyl]-6,7,10,11-tetrahydr...)
Affinity DataIC50: 743nMpH: 7.5 T: 2°CAssay Description:In vitro PDK1 assay using purified enzyme, was incubated with substrate PDKtide, and test compounds in the presence of ATP/ [gamma-32P] ATP. 32P inco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2007
Entry Details Article
PubMed