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Found 2 Enz. Inhib. hit(s) with Target = '4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase FUT5' and Ligand = 'BDBM50101904'
Target4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase FUT5(Homo sapiens (Human))
Technische Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50101904(CHEMBL52741 | GDP-Azasugar analogue)
Affinity DataIC50:  4.50E+4nMAssay Description:Inhibition of GnRH-stimulated luteinizing hormone (LH) release in rat pituitary cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase FUT5(Homo sapiens (Human))
Technische Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50101904(CHEMBL52741 | GDP-Azasugar analogue)
Affinity DataIC50:  8.20E+4nMAssay Description:Inhibitory activity against fucosyltransferase (FucT V) in the presence of 10 mM fucosyl acceptor N-acetyllactosamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed