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Found 3 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 1A' and Ligand = 'BDBM50054398'
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50054398(2-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-tetr...)
Affinity DataKi:  31nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor of rat cerebral cortex using [3H]8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50054398(2-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-tetr...)
Affinity DataKi:  31.7nMAssay Description:Binding affinity towards rat 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50054398(2-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-tetr...)
Affinity DataKi:  32nMAssay Description:Binding affinity at 5-hydroxytryptamine 1A receptor in rat cerebral cortex membranes by [3H]-8-OH-DPAT displacement.More data for this Ligand-Target Pair
In DepthDetails Article