Found 3 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 1B' and Ligand = 'BDBM50246936'
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Virginia Commonwealth University
Curated by ChEMBL
Virginia Commonwealth University
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Inhibitory activity against 5-hydroxytryptamine 1B receptor of rat striatal membrane homogenate using [3H]5-HT as the radioligand.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Virginia Commonwealth University
Curated by ChEMBL
Virginia Commonwealth University
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Binding affinity (Ki) to rat cortical membranes at 5-HT1B binding site by using [125 I] ICYP as a radioligand.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Medical College Of Virginia/Virginia Commonwealth University
Curated by ChEMBL
Medical College Of Virginia/Virginia Commonwealth University
Curated by ChEMBL
Affinity DataKi: 4.10E+3nMAssay Description:Agonist activity to the human recombinant 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair