Found 8 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 2A' and Ligand = 'BDBM50144841'
Affinity DataKi: 32nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2A receptor using displacement of [3H]5-HTMore data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Functional activity against human 5-hydroxytryptamine 2C receptor expressed in CHO cells using fluorometricimaging plate readerMore data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Displacement of [125I]DOI from human 5HT2AMore data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Displacement of [3H]5-HT from human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Agonist activity at human 5HT2A receptor expressed in HEK293 cells assessed as intracellular IP3 accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 400nMAssay Description:Agonist activity at human cloned 5HT2A receptor expressed in CHO cells assessed as myo-[3H]inositol hydrolysisMore data for this Ligand-Target Pair
Affinity DataEC50: 131nMAssay Description:Functional activity against human 5-hydroxytryptamine 2A receptor expressed in CHO cells using fluorometricimaging plate readerMore data for this Ligand-Target Pair
Affinity DataEC50: 131nMAssay Description:Binding to human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair