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Found 6 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 2A' and Ligand = 'BDBM85099'
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM85099(CAS_141474-54-6 | SDZ SER 082 FUMARATE | SDZ SER-0...)
Affinity DataKi:  245nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM85099(CAS_141474-54-6 | SDZ SER 082 FUMARATE | SDZ SER-0...)
Affinity DataKi:  331nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM85099(CAS_141474-54-6 | SDZ SER 082 FUMARATE | SDZ SER-0...)
Affinity DataKi:  513nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM85099(CAS_141474-54-6 | SDZ SER 082 FUMARATE | SDZ SER-0...)
Affinity DataKi:  631nMAssay Description:Binding affinity analysed on 5-HT 2A in rat stomach fundus.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM85099(CAS_141474-54-6 | SDZ SER 082 FUMARATE | SDZ SER-0...)
Affinity DataKd:  2.00E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 3 receptor in membranes of N1E-115 neuroblastoma cells using [3H]-ICS 205-930; Not determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM85099(CAS_141474-54-6 | SDZ SER 082 FUMARATE | SDZ SER-0...)
Affinity DataKd:  631nMAssay Description:Binding affinity towards 5-hydroxytryptamine 3 receptor in membranes of N1E-115 neuroblastoma cells using [3H]-ICS 205-930More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed