Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 2B' and Ligand = 'BDBM50144840'
Target5-hydroxytryptamine receptor 2B(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144840(CHEMBL309760 | (S)-2-(6-Bromo-2,3-dihydro-indol-1-...)
Affinity DataEC50:  11nMAssay Description:Functional activity against human 5-hydroxytryptamine 2B receptor expressed in CHO cells using fluorometric imaging plate readerMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144840(CHEMBL309760 | (S)-2-(6-Bromo-2,3-dihydro-indol-1-...)
Affinity DataKi:  30.2nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144840(CHEMBL309760 | (S)-2-(6-Bromo-2,3-dihydro-indol-1-...)
Affinity DataKi:  46nMAssay Description:Affinity for human 5-hydroxytryptamine 2B receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed