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Found 7 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 6' and Ligand = 'BDBM50073056'
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50073056(4-Bromo-N-[4-methoxy-3-(4-methyl-piperazin-1-yl)-p...)
Affinity DataKi:  2.82nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(RAT)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50073056(4-Bromo-N-[4-methoxy-3-(4-methyl-piperazin-1-yl)-p...)
Affinity DataKi:  4.79nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50073056(4-Bromo-N-[4-methoxy-3-(4-methyl-piperazin-1-yl)-p...)
Affinity DataKi:  5nMAssay Description:Antagonist activity at human recombinant 5HT6 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50073056(4-Bromo-N-[4-methoxy-3-(4-methyl-piperazin-1-yl)-p...)
Affinity DataKi:  5nMAssay Description:Binding affinity towards human 5-hydroxytryptamine 6 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50073056(4-Bromo-N-[4-methoxy-3-(4-methyl-piperazin-1-yl)-p...)
Affinity DataKi:  5nMAssay Description:Binding affinity against 5 Hydroxy tryptamine 6 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(MOUSE)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50073056(4-Bromo-N-[4-methoxy-3-(4-methyl-piperazin-1-yl)-p...)
Affinity DataKi:  22.9nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50073056(4-Bromo-N-[4-methoxy-3-(4-methyl-piperazin-1-yl)-p...)
Affinity DataIC50:  16nMAssay Description:Inhibition of human recombinant 5HT6 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed