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Found 2 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 6' and Ligand = 'BDBM50300672'
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50300672(2-(6-{[(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)su...)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT6 receptor expressed in HEK293 cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50300672(2-(6-{[(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)su...)
Affinity DataIC50:  238nMAssay Description:Antagonist activity at human 5HT6 receptor expressed in HEK293F cells assessed as inhibition of 5HT-stimulated cAMP production after 30 mins by HTRF ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed