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Found 4 Enz. Inhib. hit(s) with Target = 'Acetylcholinesterase' and Ligand = 'BDBM19126'
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Cnrs

LigandPNGBDBM19126((1R,3R,6R,7S,8R,10S,11S,14R,15R,20S)-18-[(2S)-buta...)
Affinity DataIC50:  2nMAssay Description:Inhibition of AChE activity was determined by the spectroscopic method of Ellman using acetylthiocholine iodide as substrate, in 96-well microtiter p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Cnrs

LigandPNGBDBM19126((1R,3R,6R,7S,8R,10S,11S,14R,15R,20S)-18-[(2S)-buta...)
Affinity DataIC50:  14nMAssay Description:Inhibition of AChE activity was determined by the spectroscopic method of Ellman using acetylthiocholine iodide as substrate, in 96-well microtiter p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Cnrs

LigandPNGBDBM19126((1R,3R,6R,7S,8R,10S,11S,14R,15R,20S)-18-[(2S)-buta...)
Affinity DataIC50:  4.37E+3nMAssay Description:Inhibition of AChE activity was determined by the spectroscopic method of Ellman using acetylthiocholine iodide as substrate, in 96-well microtiter p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
Cnrs

LigandPNGBDBM19126((1R,3R,6R,7S,8R,10S,11S,14R,15R,20S)-18-[(2S)-buta...)
Affinity DataIC50:  6.49E+3nMAssay Description:Inhibition of AChE activity was determined by the spectroscopic method of Ellman using acetylthiocholine iodide as substrate, in 96-well microtiter p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed